SCHEMBL7362301

SCHEMBL7362301

COC(=O)C[C@H]1C(=O)N(OC(C)=O)CCN1C(=O)C(CC(=O)N1CCN(c2ccncc2)CC1)NS(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.39
LMNA P02545 3/20 0.39
GAA P10253 2/20 0.39
ITGB3 P05106 2/20 0.39
ITGA2B P08514 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HBB P68871 1/20 0.39
TP53 P04637 2/20 0.37
ALDH1A1 P00352 4/20 0.37
PKM P14618 1/20 0.36
RAB9A P51151 1/20 0.36
MAPT P10636 3/20 0.36
P2RX7 Q99572 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
HPGD P15428 1/20 0.34
HTR7 P34969 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7935179 0.88 ITGB3 (0.40) SMN1; SMN2LMNAGAAITGB3ITGA2B
SCHEMBL7935170 0.88 ITGB3 (0.40) SMN1; SMN2LMNAGAAITGB3ITGA2B
SCHEMBL7362297 0.88 ITGB3 (0.40) SMN1; SMN2LMNAGAAITGB3ITGA2B
SCHEMBL7362643 0.88 MC4R (0.37) SMN1; SMN2LMNAKMT2ATP53ALDH1A1
Hydrochloric Acid SCHEMBL7362335 0.87 MC4R (0.37) SMN1; SMN2LMNAKMT2ATP53ALDH1A1
SCHEMBL7367999 0.84 ALDH1A1 (0.39) SMN1; SMN2LMNAGAAITGB3ITGA2B
SCHEMBL7370704 0.83 CYP2D6 (0.38) GAAITGB3ITGA2BTP53ALDH1A1
SCHEMBL7365561 0.82 GFER (0.36) GAAITGB3ITGA2BMEN1KMT2A
SCHEMBL7362706 0.81 ALDH1A1 (0.43) SMN1; SMN2LMNAGAAITGB3ITGA2B
Hydrochloric Acid SCHEMBL7935197 0.80 ALDH1A1 (0.42) SMN1; SMN2LMNAGAAITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed