SCHEMBL7362643

SCHEMBL7362643

COC(=O)C[C@H]1C(=O)N(OC(C)=O)CCN1C(=O)C(CC(=O)N1CCN(c2ccncc2)CC1)NC(=O)c1ccc(F)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.37
MC3R P41968 1/20 0.37
MC1R Q01726 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
LDHA P00338 1/20 0.34
KDM1A O60341 7/20 0.34
F10 P00742 2/20 0.33
LMNA P02545 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7362335 0.99 MC4R (0.37) MC4RMC3RMC1RSMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL7371045 0.92 ALDH1A1 (0.39) ALDH1A1MAPTLDHAKDM1AF10
SCHEMBL7362301 0.88 SMN1; SMN2 (0.39) SMN1; SMN2ALDH1A1MAPTLMNAKMT2A
SCHEMBL7362645 0.87 ITGB3 (0.47) MC4RMC3RMC1RSMN1; SMN2ALDH1A1
SCHEMBL7362639 0.87 ITGB3 (0.47) MC4RMC3RMC1RSMN1; SMN2ALDH1A1
SCHEMBL7937537 0.87 ITGB3 (0.47) MC4RMC3RMC1RSMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL7924926 0.87 ITGB3 (0.47) MC4RMC3RMC1RSMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL7362338 0.87 ITGB3 (0.47) MC4RMC3RMC1RSMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL7362333 0.87 ITGB3 (0.47) MC4RMC3RMC1RSMN1; SMN2ALDH1A1
SCHEMBL7370704 0.84 CYP2D6 (0.38) ALDH1A1MAPTHRH3TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed