SCHEMBL7365561

SCHEMBL7365561

COC(=O)C[C@H]1C(=O)N(OC(C)=O)CCN1C(=O)C(CC(=O)N1CCN(c2ccncc2)CC1)NCc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GFER P55789 2/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
MAPK1 P28482 1/20 0.36
ENPP2 Q13822 1/20 0.35
ITGB3 P05106 2/20 0.34
ITGA2B P08514 2/20 0.34
POLB P06746 1/20 0.34
GRM5 P41594 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
TGM2 P21980 1/20 0.34
TMPRSS11D O60235 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7934109 0.88 ITGB3 (0.42) GFERITGB3ITGA2BPOLB
SCHEMBL7365564 0.88 ITGB3 (0.42) GFERITGB3ITGA2BPOLB
SCHEMBL7365560 0.88 ITGB3 (0.42) GFERITGB3ITGA2BPOLB
SCHEMBL7367244 0.86 RORC (0.36) GRM5CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL7370704 0.85 CYP2D6 (0.38) GAAMAPTITGB3ITGA2BGRM5
SCHEMBL7362643 0.83 MC4R (0.37) MAPTPOLBTSHRKMT2AALDH1A1
SCHEMBL7369431 0.83 L3MBTL1 (0.34) GFERGAAMAPTCYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7362335 0.82 MC4R (0.37) MAPTPOLBTSHRKMT2AALDH1A1
Hydrochloric Acid SCHEMBL7371045 0.82 ALDH1A1 (0.39) GFERGAAMAPTMAPK1CYP3A4
SCHEMBL7362301 0.82 SMN1; SMN2 (0.39) GAAMAPTALOX15MAPK1ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed