SCHEMBL7362431

SCHEMBL7362431

NC(=O)C1CCCC1C(N)=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 4/20 0.59
PSEN1 P49768 4/20 0.47
PSEN2 P49810 4/20 0.47
APH1B Q8WW43 4/20 0.47
NCSTN Q92542 4/20 0.47
APH1A Q96BI3 4/20 0.47
PSENEN Q9NZ42 4/20 0.47
GRM4 Q14833 1/20 0.42
PEPD P12955 1/20 0.41
KMT2A Q03164 2/20 0.37
ALOX5 P09917 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
ATM Q13315 1/20 0.37
CYP2D6 P10635 1/20 0.37
GLI1 P08151 1/20 0.37
NOS2 P35228 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2343227 1.00 EPHX1 (0.59) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL1570434 0.93 EPHX1 (0.67) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL9800227 0.93 EPHX1 (0.67) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL17205447 0.93 EPHX1 (0.67) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL13557474 0.93 EPHX1 (0.67) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL9800070 0.93 EPHX1 (0.67) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL8411453 0.89 PEPD (0.56) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL7761683 0.89 PEPD (0.56) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL8411456 0.89 PEPD (0.56) EPHX1PSEN1PSEN2APH1BNCSTN
SCHEMBL7761680 0.89 PEPD (0.56) EPHX1PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114213313-B Preparation method of 1, 2-cyclopentanediimide 内蒙古源宏精细化工有限公司 2023-11-14 CN claimed
CN-115232058-A Synthesis method of gliclazide intermediate 1,2-cyclopentanedicarboxamide 上海巽田科技股份有限公司 2022-10-25 CN claimed
CN-114213313-A Preparation method of 1, 2-cyclopentadiimide 内蒙古源宏精细化工有限公司 2022-03-22 CN claimed
CN-109206358-B Synthesis method of 1, 2-cyclopentadiimide 济南爱思医药科技有限公司 2021-10-29 CN claimed
CN-112851563-A Synthesis process of N-amino-3-azabicyclo [3,3,0] octane hydrochloride 安徽金鼎医药股份有限公司 2021-05-28 CN claimed
CN-112624958-A Synthetic method of medical intermediate 1, 2-cyclopentadienimide 安徽金鼎医药股份有限公司 2021-04-09 CN claimed
US-20260085034-A1 N-(BENZHYDRYL)CYCLOALKYLCARBOXAMIDE DERIVATIVES AS INHIBITORS OF GLYCOGEN SYNTHASE 1 (GYS1) AND METHODS OF USE THEREOF HERCULES CAPITAL, INC., AS AGENT 2026-03-26 US disclosed
EP-4587422-A1 N-(BENZHYDRYL)CYCLOALKYLCARBOXAMIDE DERIVATIVES AS INHIBITORS OF GLYCOGEN SYNTHASE 1 (GYS1) AND METHODS OF USE THEREOF Maze Therapeutics, Inc. (US) 2025-07-23 EP disclosed
CN-118002062-A Reaction device and method for producing 1, 2-cyclopentadiformyl imine 浙江工业大学 2024-05-10 CN disclosed
WO-2024059661-A1 N-(BENZHYDRYL)CYCLOALKYLCARBOXAMIDE DERIVATIVES AS INHIBITORS OF GLYCOGEN SYNTHASE 1 (GYS1) AND METHODS OF USE THEREOF MAZE THERAPEUTICS, INC. (US) 2024-03-21 WO disclosed
CN-117510394-A Preparation method of N-amino-3-azabicyclo [3, 0] octane hydrochloride 内蒙古源宏精细化工有限公司 2024-02-06 CN disclosed
CN-117510394-A Preparation method of N-amino-3-azabicyclo [3, 0] octane hydrochloride 内蒙古源宏精细化工有限公司 2024-02-06 CN disclosed
CN-115232057-B Synthesis method of gliclazide intermediate 3-azabicyclo [3.3.0] octane 上海巽田科技股份有限公司 2024-01-26 CN disclosed
CN-103183632-A Purification method of 3-azabicyclo-octane hydrochloride SHANDONG FANGMING PHARM GROUP 2013-07-03 CN disclosed
CN-102850257-A Preparation method of 1,2-cyclopentane dicarboximide SHANDONG FANGMING PHARM GROUP 2013-01-02 CN disclosed
CN-102850257-A Preparation method of 1,2-cyclopentane dicarboximide SHANDONG FANGMING PHARM GROUP 2013-01-02 CN disclosed
CN-100424077-C Cyclopentane1,2-diimide preparation method TAIZHOU SIWEI CHEMICAL PLANT (CN) 2008-10-08 CN disclosed
CN-1876636-A Cyclopentane1,2-diimide preparation method TAIZHOU SIWEI CHEMICAL PLANT (CN) 2006-12-13 CN disclosed
EP-1087937-A1 CYCLIC HYDROXAMIC ACIDS AS METALLOPROTEINASE INHIBITORS Du Pont Pharmaceuticals Company (US) 2001-04-04 EP disclosed
WO-1999065867-A1 CYCLIC HYDROXAMIC ACIDS AS METALLOPROTEINASE INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 1999-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260085034-A1 N-(BENZHYDRYL)CYCLOALKYLCARBOXAMIDE DERIVATIVES AS INHIBITORS OF GLYCOGEN SYNTHASE 1 (GYS1) AND METHODS OF USE THEREOF GYS2, GYS1, PYGL EPHX1 2283/4885PSEN1 97/4885PSEN2 184/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.