SCHEMBL7362444

SCHEMBL7362444

C=CC(=O)C(C)Cc1ccc(F)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.39
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
RIPK1 Q13546 1/20 0.38
DPP7 Q9UHL4 1/20 0.37
PIN1 Q13526 1/20 0.36
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
DPP8 Q6V1X1 1/20 0.34
MME P08473 1/20 0.34
ACE P12821 1/20 0.34
CPA1 P15085 1/20 0.34
ACE2 Q9BYF1 1/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
SLC6A2 P23975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9227299 0.82 TRPA1 (0.47) CPA1
SCHEMBL6003677 0.80 TBXAS1 (0.44) DPP4MAOAMAOBRIPK1PIN1
SCHEMBL6005325 0.80 TBXAS1 (0.44) DPP4MAOAMAOBRIPK1PIN1
SCHEMBL6003686 0.80 TBXAS1 (0.44) DPP4MAOAMAOBRIPK1PIN1
SCHEMBL31067929 0.80 TBXAS1 (0.44) DPP4MAOAMAOBRIPK1PIN1
SCHEMBL7360275 0.80 SLC1A1 (0.48) MAOAMAOB
SCHEMBL6400128 0.79 DPP4 (0.44) DPP4MAOAMAOBRIPK1DPP7
SCHEMBL27952958 0.78 MAOA (0.39) DPP4MAOAMAOBRIPK1DPP7
SCHEMBL23030411 0.76 MAOA (0.42) DPP4MAOAMAOBPIN1MME
SCHEMBL21400126 0.76 DPP4 (0.39) DPP4MAOAMAOBRIPK1DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112269-A2 HIV PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-07-04 EP disclosed
WO-2000015634-A2 HIV PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2000-03-23 WO disclosed