SCHEMBL7362579

SCHEMBL7362579

C=CCn1ccnc1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
ADORA2B P29275 1/20 0.32
ARG1 P05089 1/20 0.32
MAP2K2 P36507 1/20 0.31
MAP2K1 Q02750 1/20 0.31
NPC1 O15118 2/20 0.31
KMT2A Q03164 2/20 0.31
TSHR P16473 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ESR1 P03372 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
MEN1 O00255 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28411111 0.84 SMN1; SMN2 (0.37) ADORA2BARG1NPC1KMT2AESR1
SCHEMBL4314338 0.77 SMN1; SMN2 (0.39) ALDH1A1ARG1NPC1KMT2ASMN1; SMN2
SCHEMBL3810263 0.77 ALDH1A1 (0.35) ALDH1A1ARG1NPC1TSHRKDM4E
SCHEMBL30554012 0.76 KMT2A (0.43) ALDH1A1NPC1KMT2AKDM4ERAB9A
SCHEMBL2719494 0.74 PPARG (0.51) ALDH1A1NPC1KDM4ESMN1; SMN2RAB9A
SCHEMBL31210326 0.74 ARG1 (0.39) ALDH1A1ARG1ESR1SMN1; SMN2RAB9A
SCHEMBL27845254 0.74 TLR8 (0.42) ALDH1A1ARG1KMT2ASMN1; SMN2
SCHEMBL4333586 0.72 SMN1; SMN2 (0.33) ALDH1A1ARG1NPC1KDM4EESR1
SCHEMBL5616672 0.72
SCHEMBL5141262 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5789406-A Indeno 1,2-E!pyrazine-4-ones, their preparation and the medicaments containing them RHONE-POULENC RORER S.A. (FR) 1998-08-04 US disclosed
US-5672705-A ANTIISCHEMIC AGENTS TREATING NERVOUS SYSTEM DISORDERS, HUNTINGTON' DISEASE, ALZHEIMER'S DISEASE, PARKINSON'S DISEASE RHONE-POULENC RORER S.A. (FR) 1997-09-30 US disclosed
EP-0726900-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS Aventis Pharma S.A. (FR) 1996-08-21 EP disclosed
WO-1995012594-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1995-05-11 WO disclosed