SCHEMBL4333586

SCHEMBL4333586

CN(C)Cn1ccnc1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ARG1 P05089 1/20 0.32
MAPT P10636 1/20 0.31
FDPS P14324 1/20 0.31
TLR8 Q9NR97 2/20 0.31
ALPL P05186 1/20 0.31
ALPI P09923 1/20 0.31
ALPG P10696 1/20 0.31
PLAA Q9Y263 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HTT P42858 1/20 0.31
CDK8 P49336 1/20 0.31
CDK19 Q9BWU1 1/20 0.31
ESR1 P03372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4327360 0.85 HTT (0.33) SMN1; SMN2ALDH1A1NPC1RAB9AARG1
SCHEMBL4314338 0.80 SMN1; SMN2 (0.39) SMN1; SMN2ALDH1A1NPC1RAB9AARG1
SCHEMBL31210326 0.77 ARG1 (0.39) SMN1; SMN2ALDH1A1RAB9AARG1TLR8
SCHEMBL27845254 0.77 TLR8 (0.42) SMN1; SMN2ALDH1A1ARG1TLR8
SCHEMBL3810263 0.77 ALDH1A1 (0.35) SMN1; SMN2ALDH1A1NPC1RAB9AARG1
SCHEMBL7362579 0.72 ALDH1A1 (0.33) SMN1; SMN2ALDH1A1NPC1RAB9AARG1
SCHEMBL18839651 0.71 KDM4E (0.44) SMN1; SMN2ALDH1A1NPC1MAPTKDM4E
SCHEMBL28205879 0.70 CYP11B1 (0.42) SMN1; SMN2ALDH1A1NPC1RAB9AKDM4E
SCHEMBL4325015 0.70 SIRT2 (0.38) ALDH1A1ARG1CDK8
SCHEMBL3313595 0.70 ALDH1A1 (0.59) SMN1; SMN2ALDH1A1NPC1RAB9AFDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009141386-A1 DERIVATIVES OF QUINOLINES AND QUINOXALINES AS PROTEIN TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2009-11-26 WO disclosed