SCHEMBL7362909

SCHEMBL7362909

CNC(CN)c1ccc(OC)c(OC2Cc3ccccc3C2)c1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.50
PDE4A P27815 13/20 0.49
PDE4D Q08499 9/20 0.49
PDE4C Q08493 7/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7144760 0.84 PDE4B (0.55) PDE4BPDE4APDE4DPDE4C
SCHEMBL7919796 0.83 PDE4B (0.61) PDE4BPDE4APDE4DPDE4C
SCHEMBL9378730 0.79 PDE4A (0.40) PDE4BPDE4APDE4DPDE4C
SCHEMBL7364925 0.77 PDE4B (0.57) PDE4BPDE4APDE4DPDE4C
SCHEMBL7356450 0.76 LMNA (0.37) PDE4BPDE4APDE4DPDE4C
SCHEMBL4727275 0.76 PDE4B (0.55) PDE4BPDE4APDE4DPDE4C
SCHEMBL4728355 0.74 PDE4B (0.56) PDE4BPDE4APDE4DPDE4C
SCHEMBL1157507 0.74 PDE4B (0.60) PDE4BPDE4APDE4DPDE4C
SCHEMBL7364049 0.74 PDE4B (0.52) PDE4BPDE4APDE4DPDE4C
SCHEMBL7360381 0.74 PDE4A (0.46) PDE4BPDE4APDE4DPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5459145-A Calcium independent camp phosphodiesterase inhibitor antidepressant PFIZER INC. (US) 1995-10-17 US disclosed
US-5294730-A A-Amino-4-alkoxy-3-polycycloalkyloxybenzyl cyanide derivatives PFIZER INC. (US) 1994-03-15 US disclosed
EP-0247725-B1 Calcium independent camp phosphodiestrerase inhibitor antidepressant PFIZER (US) 1994-03-02 EP disclosed
US-5196426-A CALCIUM INDEPENDENT C AMP PHOSPHODIESTERASE INHIBITOR ANTIDEPRESSANT PFIZER INC. (US) 1993-03-23 US disclosed
US-5128358-A Aryl substituted nitrogen heterocyclic antidepressants PFIZER INC. (US) 1992-07-07 US disclosed
EP-0247725-A2 Calcium independent camp phosphodiestrerase inhibitor antidepressant PFIZER INC. (US) 1987-12-02 EP disclosed
WO-1987006576-A1 CALCIUM INDEPENDENT CAMP PHOSPHODIESTERASE INHIBITOR ANTIDEPRESSANT PFIZER INC. (US) 1987-11-05 WO disclosed