SCHEMBL7363206

SCHEMBL7363206

CN(C)c1ncccc1NC(=NC#N)NCCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPK1 P28482 2/20 0.43
ALOX12 P18054 4/20 0.39
CYP1A2 P05177 3/20 0.37
CYP3A4 P08684 3/20 0.37
CYP2D6 P10635 3/20 0.37
CYP2C19 P33261 3/20 0.37
LMNA P02545 2/20 0.37
CYP2C9 P11712 2/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HPGD P15428 2/20 0.37
P2RX7 Q99572 2/20 0.37
SLC2A1 P11166 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360081 0.83 RAB9A (0.46) ALDH1A1RAB9ASMN1; SMN2KDM4EMAPK1
SCHEMBL7359999 0.79 P2RX7 (0.52) ALDH1A1RAB9ASMN1; SMN2KDM4EMAPK1
SCHEMBL7363209 0.78 NAMPT (0.48) KDM4EALOX12CYP1A2CYP3A4CYP2D6
SCHEMBL7363204 0.77 P2RX7 (0.42) ALDH1A1RAB9AMAPK1LMNAHPGD
SCHEMBL8622514 0.77 P2RX7 (0.42) ALDH1A1RAB9AMAPK1LMNAHPGD
SCHEMBL8622507 0.77 P2RX7 (0.42) ALDH1A1RAB9AMAPK1LMNAHPGD
SCHEMBL7361542 0.74 HTT (0.34) P2RX7HTT
SCHEMBL7361539 0.74 HTT (0.34) P2RX7HTT
SCHEMBL9149002 0.74 BCL6 (0.62) RAB9ASMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL8625066 0.73 HTT (0.39) ALDH1A1RAB9ASMN1; SMN2KDM4EALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741708-A1 CYANOGUANIDINES AS K-CHANNEL BLOCKERS PHARMACIA & UPJOHN COMPANY (US) 1996-11-13 EP claimed
WO-1995020579-A1 CYANOGUANIDINES AS K-CHANNEL BLOCKERS PHARMACIA & UPJOHN COMPANY (US) 1995-08-03 WO claimed