SCHEMBL7363209

SCHEMBL7363209

CN(C)c1ncccc1NC(=NCCc1ccccc1)NC#N

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.48
P2RX7 Q99572 7/20 0.44
QPCT Q16769 2/20 0.39
HRH4 Q9H3N8 3/20 0.38
HRH2 P25021 2/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
PKM P14618 1/20 0.37
ALOX12 P18054 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360003 0.79 P2RX7 (0.61) NAMPTP2RX7QPCTHRH4HRH2
SCHEMBL7363206 0.78 ALDH1A1 (0.43) P2RX7KDM4ELMNACYP1A2POLB
SCHEMBL8622511 0.77 P2RX7 (0.69) P2RX7LMNACYP1A2CYP3A4CYP2C9
SCHEMBL7361546 0.74 P2RX7 (0.40) P2RX7HTT
SCHEMBL7350535 0.74 NAMPT (0.62) NAMPTP2RX7QPCTHRH4HRH2
SCHEMBL7423091 0.71 NAMPT (0.59) NAMPTP2RX7QPCTHRH4HRH2
SCHEMBL9148294 0.70 HRH4 (0.50) NAMPTQPCTHRH4HRH2
SCHEMBL9838248 0.69 NAMPT (0.57) NAMPTP2RX7QPCTHRH4HRH2
SCHEMBL7424829 0.68 HRH4 (0.53) NAMPTQPCTHRH4HRH2
SCHEMBL7363204 0.68 P2RX7 (0.42) P2RX7LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741708-A1 CYANOGUANIDINES AS K-CHANNEL BLOCKERS PHARMACIA & UPJOHN COMPANY (US) 1996-11-13 EP claimed
WO-1995020579-A1 CYANOGUANIDINES AS K-CHANNEL BLOCKERS PHARMACIA & UPJOHN COMPANY (US) 1995-08-03 WO claimed