SCHEMBL7363525

SCHEMBL7363525

COC(=O)[C@H](Cc1ccc([N+](=O)[O-])cc1)N(C(=O)OCc1ccccc1)C(=O)[C@@H](N)C(C)C

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ITGA4 P13612 1/20 0.43
ITGB7 P26010 1/20 0.43
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
TP53 P04637 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CTSL P07711 2/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MC4R P32245 1/20 0.41
HTR2A P28223 1/20 0.39
LTA4H P09960 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8588884 0.92 MEN1 (0.43) MEN1KMT2AITGA4ITGB7RAB9A
SCHEMBL30841321 0.81 ITGA4 (0.46) MEN1KMT2AITGA4ITGB7RAB9A
SCHEMBL8590776 0.79 SLC15A1 (0.45) MEN1KMT2ARAB9ANPC1LTA4H
SCHEMBL2388059 0.77 CTSL (0.49) MEN1KMT2AITGA4ITGB7CTSL
SCHEMBL6904576 0.77 ABCB1 (0.47) ALDH1A1LTA4H
SCHEMBL9330125 0.77 ABCB1 (0.47) ALDH1A1LTA4H
SCHEMBL7281801 0.75 MEN1 (0.52) MEN1KMT2AITGA4ITGB7RAB9A
SCHEMBL9706834 0.74 MC4R (0.51) MEN1KMT2AITGA4ITGB7RAB9A
SCHEMBL1151902 0.73 CTSB (0.46) MEN1KMT2AALDH1A1LTA4H
SCHEMBL9023544 0.73 SLC15A1 (0.45) MEN1KMT2ACTSLALDH1A1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998038990-A1 METHOD OF TREATING TRAUMA ASSOCIATED WITH BRAIN, SPINAL CORD OR PERIPHERAL NERVE INJURY USING CARBOBENZYLOXY N-PROTECTED DI- AND TRIPEPTIDE PHENYLALANINALS HOECHST MARION ROUSSEL, INC. (US) 1998-09-11 WO disclosed
EP-0802909-A2 SUBSTITUTED OXAZOLIDINE CALPAIN AND/OR CATHEPSIN B INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1997-10-29 EP disclosed
WO-1996021655-A2 SUBSTITUTED OXAZOLIDINE CALPAIN AND/OR CATHEPSIN B INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1996-07-18 WO disclosed