SCHEMBL7363736

SCHEMBL7363736

COc1cc([C]=O)ccc1N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.55
CYP3A4 P08684 4/20 0.55
TDP1 Q9NUW8 4/20 0.55
TSHR P16473 1/20 0.55
HSD17B10 Q99714 1/20 0.55
HTT P42858 2/20 0.50
APP P05067 3/20 0.44
ADRA2B P18089 1/20 0.43
PTGS1 P23219 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.39
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
IDO1 P14902 1/20 0.38
THRB P10828 1/20 0.38
S100B P04271 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10567689 0.84 ALDH1A1 (0.53) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL29559790 0.82 ALDH1A1 (0.57) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL220780 0.82 ALDH1A1 (0.57) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL56335 0.81 CA2 (0.48) ALDH1A1CYP3A4TDP1TSHRPOLB
SCHEMBL17729353 0.80 ALDH1A1 (0.55) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL22146862 0.80 ALDH1A1 (0.55) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL27701508 0.78 APP (0.60) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL11593518 0.78 ALDH1A1 (0.39) ALDH1A1CYP3A4TDP1HPGD
SCHEMBL2123029 0.78 AR (0.44) ALDH1A1CYP3A4TDP1GAAHPGD
SCHEMBL5125769 0.76 LMNA (0.40) ALDH1A1CYP3A4TDP1HTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100339442-C Method for preparing organic pigment of red benzimidazolones UNIV HUADONG TECHNOLOGY (CN) 2007-09-26 CN claimed
CN-1563202-A Method for preparing organic pigment of red benzimidazolones UNIV HUADONG TECHNOLOGY (CN) 2005-01-12 CN claimed
EP-3099694-A1 COMPOUNDS GlaxoSmithKline Intellectual Property Development Limited (GB) 2016-12-07 EP disclosed
WO-2015113451-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2015-08-06 WO disclosed
CN-100339442-C Method for preparing organic pigment of red benzimidazolones UNIV HUADONG TECHNOLOGY (CN) 2007-09-26 CN disclosed
CN-1563202-A Method for preparing organic pigment of red benzimidazolones UNIV HUADONG TECHNOLOGY (CN) 2005-01-12 CN disclosed
WO-1998050030-A1 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIVERSITY OF PITTSBURGH (US) 1998-11-12 WO disclosed
EP-0846127-A1 ACYLATED OLIGOPEPTIDE DERIVATIVES HAVING CELL SIGNAL INHIBITING ACTIVITY Novartis AG (CH) 1998-06-10 EP disclosed
WO-1997008193-A1 ACYLATED OLIGOPEPTIDE DERIVATIVES HAVING CELL SIGNAL INHIBITING ACTIVITY NOVARTIS AG (CH) 1997-03-06 WO disclosed
WO-1997007131-A1 ACYLATED OLIGOPEPTIDES CONTAINING PHOSPHOTYROSINE AS INHIBITORS OF PROTEIN TYROSINE KINASES NOVARTIS AG (CH) 1997-02-27 WO disclosed