SCHEMBL7363869

SCHEMBL7363869

Cc1ccc(F)c(N)c1.Cc1ccc(F)c(O)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
ALOX15 P16050 2/20 0.57
HSD17B10 Q99714 1/20 0.57
TDP1 Q9NUW8 3/20 0.46
TP53 P04637 2/20 0.46
CYP3A4 P08684 2/20 0.46
TRPA1 O75762 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
THRB P10828 1/20 0.46
CA3 P07451 1/20 0.45
CA6 P23280 1/20 0.45
CA5A P35218 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
CA5B Q9Y2D0 1/20 0.45
CA1 P00915 1/20 0.41
HSD17B14 Q9BPX1 1/20 0.40
LMNA P02545 2/20 0.39
CHRM1 P11229 1/20 0.39
SLC6A2 P23975 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30413683 0.87
SCHEMBL59217 0.87
SCHEMBL12127 0.87
SCHEMBL28749668 0.79 TDP1 (0.50) ALDH1A1ALOX15HSD17B10TDP1TP53
SCHEMBL27816817 0.76 TRPA1 (0.46) ALDH1A1ALOX15HSD17B10TDP1TP53
SCHEMBL27870665 0.76 TRPA1 (0.46) ALDH1A1ALOX15HSD17B10TDP1TP53
Metacresol SCHEMBL10549611 0.74 ACHE (0.65) ALDH1A1ALOX15HSD17B10TDP1TP53
SCHEMBL33821 0.73
SCHEMBL4866842 0.73 ALOX15 (0.65) ALDH1A1ALOX15HSD17B10TDP1TP53
SCHEMBL29356215 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0538384-A4 OXAMIDES SMITHKLINE BEECHAM CORP (US) 1995-04-12 EP disclosed
US-5393788-A Phenylalkyl oxamides SMITHKLINE BEECHAM CORPORATION (US) 1995-02-28 US disclosed
EP-0538384-A1 OXAMIDES SMITHKLINE BEECHAM CORPORATION (US) 1993-04-28 EP disclosed
WO-1992000968-A1 OXAMIDES SMITHKLINE BEECHAM CORPORATION (US) 1992-01-23 WO disclosed