SCHEMBL7364147

SCHEMBL7364147

CCCCS(=O)(=O)CC(CS(=O)(=O)CCCC)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCLC P48506 1/20 0.53
CA2 P00918 2/20 0.47
MAPK1 P28482 1/20 0.47
CHRM1 P11229 1/20 0.43
AKR1A1 P14550 1/20 0.43
CHRM3 P20309 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43
DRD3 P35462 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SLC1A2 P43004 2/20 0.40
SLC1A1 P43005 2/20 0.40
SLC1A3 P43003 1/20 0.40
GRIK1 P39086 2/20 0.39
GRIK2 Q13002 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1376126 0.86 GCLC (0.49) GCLCCA2MAPK1
SCHEMBL7361066 0.79 CA1 (0.52) GCLCCA2HDAC1HDAC2FAAH
SCHEMBL6906378 0.76 ACE2 (0.47) GCLCCA2FAAHCES2CES1
SCHEMBL9067216 0.75 NOS2 (0.54) GCLCCA2SLC1A2SLC1A1SLC1A3
SCHEMBL6671787 0.75 FAAH (0.42) GCLCCA2FAAHCES2CES1
SCHEMBL7054608 0.74 FOLH1 (0.47) GCLCCA2MAPK1CHRM1AKR1A1
SCHEMBL1374895 0.73 GCLC (0.51) GCLCCHRM1AKR1A1CHRM3HTR2A
SCHEMBL6646261 0.73 NOS2 (0.53) GCLCCA2SLC1A2SLC1A1SLC1A3
Hydrochloric Acid SCHEMBL9359667 0.73 ACE2 (0.49) CA2FAAHCES2CES1GPR84
SCHEMBL2303290 0.73 CA2 (0.41) CA2MAPK1FAAHCES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235928-B1 ENZYME INHIBITOR MATRIX METALLOPROTEINASE FAMILY, INCLUDING COLLAGENASE, STROMELYSIN, AND GELATINASE, THE COMPOUNDS OR PHARMACEUTICAL COMPOSITIONS PHARMACIA & UPJOHN COMPANY 2001-05-22 US disclosed
EP-0929519-A1 $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 1999-07-21 EP disclosed
US-5847153-A β-sulfonyl hydroxamic acids PHARMACIA & UPJOHN COMPANY (US) 1998-12-08 US disclosed
WO-1998013340-A1 β-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 1998-04-02 WO disclosed