SCHEMBL7364338

SCHEMBL7364338

NC(=O)C[C@H](NC(=O)c1ccc2ccccc2n1)C(=O)NNC[C@H](O)CCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.49
HDAC1 Q13547 2/20 0.45
CYP3A4 P08684 3/20 0.45
OPRM1 P35372 2/20 0.45
OPRK1 P41145 2/20 0.45
ABCC3 O15438 1/20 0.45
ABCC4 O15439 1/20 0.45
CACNA1F O60840 1/20 0.45
ABCB11 O95342 1/20 0.45
ABCB1 P08183 1/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
TACR2 P21452 1/20 0.45
TBXAS1 P24557 1/20 0.45
DRD3 P35462 1/20 0.45
AVPR1A P37288 1/20 0.45
OPRD1 P41143 1/20 0.45
HTR2B P41595 1/20 0.45
CACNA1D Q01668 1/20 0.45
SLC6A3 Q01959 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8735281 1.00 CTSD (0.49) CTSDHDAC1CYP3A4OPRM1OPRK1
SCHEMBL8842831 0.83 CTSD (0.52) CTSDHDAC1CYP3A4OPRM1OPRK1
SCHEMBL8735285 0.81 CTSD (0.45) CTSDHDAC1CYP3A4OPRM1OPRK1
SCHEMBL8732141 0.81 CTSD (0.47) CTSDHDAC1CYP3A4OPRM1OPRK1
SCHEMBL8731972 0.77 MMP3 (0.49)
SCHEMBL6444839 0.77 ALDH1A1 (0.58) CTSDHDAC1ALDH1A1TP53GAA
SCHEMBL561849 0.77 ALDH1A1 (0.58) CTSDHDAC1ALDH1A1TP53GAA
SCHEMBL8734194 0.77 CYP3A4 (0.55) CTSDHDAC1CYP3A4OPRM1OPRK1
Hydrochloric Acid SCHEMBL4862500 0.76 ALDH1A1 (0.57) CTSDHDAC1ALDH1A1TP53GAA
SCHEMBL7277774 0.76 CTSD (0.57) CTSDHDAC1CYP3A4OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602175-A HYDROXYETHYLAMINE COMPOUNDS; USEFUL IN TREATMENT OF INFECTIONS CAUSED BY THE HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1997-02-11 US disclosed
EP-0558673-B1 RETROVIRAL PROTEASE INHIBITORS MONSANTO CO (US) 1996-04-17 EP disclosed
US-5482947-A ENZYME INHIBITORS FOR HIV PROTEASE INHIBITION FROM UREA OR THIOUREA COMPOUNDS TALLEY JOHN J (US) 1996-01-09 US disclosed
EP-0558603-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1993-09-08 EP disclosed
WO-1992008688-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1992-05-29 WO disclosed