SCHEMBL8731972

SCHEMBL8731972

NC(=O)C[C@@H](NC(=O)OCc1ccccc1)C(=O)NNCC(O)CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 1/20 0.49
PSMB1 P20618 1/20 0.48
CTSL P07711 7/20 0.48
CTSK P43235 2/20 0.47
TACR1 P25103 1/20 0.47
CASP1 P29466 3/20 0.46
MME P08473 1/20 0.46
ECE1 P42892 1/20 0.46
PSMB8 P28062 1/20 0.45
PSMB5 P28074 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8731991 0.80 PSMB1 (0.46) MMP3PSMB1CTSLCTSKCASP1
SCHEMBL9064404 0.79 CTSL (0.50) MMP3PSMB1CTSLCASP1MME
SCHEMBL18735868 0.78 PSMB1 (0.56) PSMB1CTSLCTSKTACR1MME
SCHEMBL11124167 0.78 MME (0.64) PSMB1CTSLCTSKTACR1MME
SCHEMBL7270223 0.78 PSMB1 (0.59) PSMB1CTSLCTSKTACR1MME
SCHEMBL722757 0.78 MME (0.62) PSMB1CTSKTACR1CASP1MME
SCHEMBL3569541 0.78 MME (0.62) PSMB1CTSKTACR1CASP1MME
SCHEMBL7688519 0.78 PSMB1 (0.57) PSMB1CTSLCTSKTACR1CASP1
SCHEMBL8955765 0.78 CTSL (0.57) PSMB1CTSLCTSKTACR1CASP1
SCHEMBL1491365 0.78 MME (0.62) PSMB1CTSKTACR1CASP1MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708004-A ENZYME INHIBITORS FOR TREATMENT OF AIDS MONSANTO COMPANY (US) 1998-01-13 US disclosed
US-5703076-A TREATING HIV, AIDS G. D. SEARLE & CO. (US) 1997-12-30 US disclosed
US-5698569-A Retroviral protease inhibitors G. D. SEARLE & CO. (US) 1997-12-16 US disclosed
US-5510349-A HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510378-A Retroviral protease inhibitors G.D. SEARLE & CO. (US) 1996-04-23 US disclosed