SCHEMBL7365263

SCHEMBL7365263

CCOC(=O)[C@H](Cc1cccnc1)NC(=O)CC1CCCN(CCc2ccncc2)C1=O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.46
ITGA2B P08514 3/20 0.46
NLRP3 Q96P20 2/20 0.40
POLB P06746 1/20 0.38
ACE P12821 3/20 0.37
FKBP1A P62942 1/20 0.37
ALDH1A1 P00352 2/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
TP53 P04637 1/20 0.36
LMNA P02545 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
YAP1 P46937 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7345393 0.87 ITGB3 (0.46) ITGB3ITGA2BNLRP3POLBACE
SCHEMBL7341598 0.85 ITGB3 (0.43) ITGB3ITGA2BNLRP3POLBACE
SCHEMBL7365261 0.82 ITGB3 (0.47) ITGB3ITGA2BFKBP1AALDH1A1TP53
SCHEMBL7342847 0.77 ITGB3 (0.44) ITGB3ITGA2BNLRP3ACEFKBP1A
SCHEMBL7342258 0.73 ITGB3 (0.45) ITGB3ITGA2BACEALDH1A1TP53
SCHEMBL7371673 0.72 ITGB3 (0.51) ITGB3ITGA2BACEALDH1A1HRH3
SCHEMBL7342693 0.71 ITGB3 (0.79) ITGB3ITGA2BACEHRH3
SCHEMBL7369685 0.71 ITGB3 (0.47) ITGB3ITGA2BFKBP1AHTT
SCHEMBL3288909 0.71 HDAC1 (0.51) ITGB3ITGA2BACE
SCHEMBL6739005 0.71 NLRP3 (0.49) NLRP3POLBALDH1A1TP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0866705-A4 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1999-03-03 EP disclosed
EP-0866705-A1 FIBRINOGEN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-09-30 EP disclosed
WO-1997014417-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-04-24 WO disclosed