SCHEMBL7365364

SCHEMBL7365364

NC(=NCl)Nc1cncc2cc(S(=O)(=O)N3CCC[C@@H]3C(=O)O)ccc12

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PLAU P00749 4/20 0.54
KDM4E B2RXH2 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 2/20 0.44
HCRTR1 O43613 7/20 0.44
HCRTR2 O43614 7/20 0.44
RECQL P46063 1/20 0.42
TSHR P16473 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CCR4 P51679 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7368609 0.99 PLAU (0.53) PLAUKDM4EHSD17B10LMNAHCRTR1
Hydrochloric Acid SCHEMBL7366142 0.99 PLAU (0.53) PLAUKDM4EHSD17B10LMNAHCRTR1
SCHEMBL7370379 0.97 PLAU (0.54) PLAUKDM4EHSD17B10LMNAHCRTR1
Hydrochloric Acid SCHEMBL7369946 0.96 PLAU (0.54) PLAUKDM4EHSD17B10LMNAHCRTR1
Hydrochloric Acid SCHEMBL7369169 0.96 PLAU (0.54) PLAUKDM4EHSD17B10LMNAHCRTR1
SCHEMBL7380965 0.94 PLAU (0.53) PLAULMNAHCRTR1HCRTR2RECQL
SCHEMBL7450926 0.91 PLAU (0.51) PLAUKDM4EHSD17B10LMNAHCRTR1
Hydrochloric Acid SCHEMBL7368466 0.90 PLAU (0.51) PLAUKDM4EHSD17B10LMNAHCRTR1
SCHEMBL7368857 0.88 LMNA (0.45) PLAUKDM4ELMNAHCRTR1HCRTR2
SCHEMBL7374254 0.87 CASP3 (0.50) PLAULMNAHCRTR1HCRTR2RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077945-A1 ISOQUINOLINES AS UROKINASE INHIBITORS PFIZER INC. (US) 2001-02-28 EP claimed
WO-2000005214-A2 ISOQUINOLINES AS UROKINASE INHIBITORS PFIZER INC. (US) 2000-02-03 WO claimed
EP-1242120-A2 COMBINATIONS OF GROWTH FACTORS AND I:UPA OR I:MMP FOR THE TREATMENT OF DAMAGED TISSUE Pfizer Limited (GB) 2002-09-25 EP disclosed
WO-2001049309-A2 COMBINATIONS OF GROWTH FACTORS AND I: UPA OR I: MMP FOR THE TREATMENT OF DAMAGED TISSUE PFIZER LIMITED (GB) 2001-07-12 WO disclosed
EP-1077945-A1 ISOQUINOLINES AS UROKINASE INHIBITORS PFIZER INC. (US) 2001-02-28 EP disclosed
WO-2000005214-A2 ISOQUINOLINES AS UROKINASE INHIBITORS PFIZER INC. (US) 2000-02-03 WO disclosed