SCHEMBL7365366

SCHEMBL7365366

CC(=O)SCC(CN[C@@H](Cc1c[nH]c2ccccc12)C(=O)O)C(=O)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.53
MEN1 O00255 4/20 0.53
PPARG P37231 1/20 0.50
ECE1 P42892 1/20 0.49
P2RY14 Q15391 1/20 0.49
ERAP2 Q6P179 3/20 0.48
LNPEP Q9UIQ6 3/20 0.48
ERAP1 Q9NZ08 2/20 0.48
POLB P06746 1/20 0.47
HTT P42858 1/20 0.47
HSP90AA1 P07900 1/20 0.47
HSP90AB1 P08238 1/20 0.47
LTA4H P09960 1/20 0.47
PLA2G2A P14555 1/20 0.47
KCNA5 P22460 1/20 0.46
IL1RN P18510 1/20 0.46
ALOX15 P16050 1/20 0.46
MMP2 P08253 1/20 0.45
MMP13 P45452 1/20 0.45
MMP14 P50281 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6169855 0.84 LTA4H (0.59) KMT2AMEN1ECE1P2RY14LTA4H
SCHEMBL7361908 0.81 ALOX15 (0.50) ECE1ERAP2ALOX15MMP2
SCHEMBL7367496 0.81 ALOX15 (0.50) ECE1ERAP2ALOX15MMP2
SCHEMBL6172199 0.75 LTA4H (0.69) ECE1LTA4HALOX15
SCHEMBL6172205 0.75 LTA4H (0.69) ECE1LTA4HALOX15
SCHEMBL7360589 0.75 CYP1A2 (0.46)
SCHEMBL11430738 0.75 ACE (0.67) ECE1LTA4HALOX15
SCHEMBL7359906 0.74 ECE1 (0.60) ECE1MMP2
SCHEMBL7430891 0.73 KDM4E (0.61) KMT2AMEN1POLBALOX15
SCHEMBL7367820 0.73 FPR2 (0.57) ECE1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888341-A1 NOVEL SULPHUR DERIVATIVES COMPRISING AN AMIDE BOND, METHOD FOR PREPARING SAME, USE THEREOF AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH DERIVATIVES HOECHST MARION ROUSSEL (FR) 1999-01-07 EP disclosed
WO-1997032874-A1 NOVEL SULPHUR DERIVATIVES COMPRISING AN AMIDE BOND, METHOD FOR PREPARING SAME, USE THEREOF AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH DERIVATIVES HOECHST MARION ROUSSEL (FR) 1997-09-12 WO disclosed