SCHEMBL7366245

SCHEMBL7366245

CC(C)(Cc1c(N)cccc1-c1ccccc1)S(N)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PTGS2 P35354 3/20 0.39
CA2 P00918 3/20 0.36
CA9 Q16790 3/20 0.36
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CYP2C9 P11712 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
NSD2 O96028 3/20 0.34
PTGS1 P23219 2/20 0.33
PTPRC P08575 1/20 0.33
ADORA2A P29274 1/20 0.33
GAA P10253 1/20 0.33
HTR6 P50406 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9275263 0.85 CA12 (0.43) ALDH1A1PTGS2CA2CA9CA12
SCHEMBL9373748 0.82 DPP4 (0.36) PTGS2CA2CA9CA12CA1
SCHEMBL7369396 0.73 NPC1 (0.38) ALDH1A1HSD17B10CA2CA9CA12
SCHEMBL17494172 0.73 ALDH1A1 (0.48) ALDH1A1HSD17B10PTGS2PTPRCADORA2A
SCHEMBL8029374 0.73 CA12 (0.38) HSD17B10PTGS2CA2CA9CA12
SCHEMBL31570105 0.72 ALDH1A1 (0.56) ALDH1A1HSD17B10GAA
SCHEMBL20263706 0.72 ALDH1A1 (0.56) ALDH1A1HSD17B10GAA
SCHEMBL29636396 0.71 ALDH1A1 (0.46) ALDH1A1HSD17B10PTGS2CA2CA9
SCHEMBL3789187 0.70 ALDH1A1 (0.58) ALDH1A1HSD17B10GAA
SCHEMBL3780645 0.70 ALDH1A1 (0.58) ALDH1A1HSD17B10CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0960102-A1 AMIDINOINDOLES, AMIDINOAZOLES, AND ANALOGS THEREOF AS INHIBITORS OF FACTOR Xa AND OF THROMBIN Du Pont Pharmaceuticals Company (US) 1999-12-01 EP disclosed
WO-1998001428-A1 AMIDINOINDOLES, AMIDINOAZOLES, AND ANALOGS THEREOF AS INHIBITORS OF FACTOR Xa AND OF THROMBIN DU PONT PHARMACEUTICALS COMPANY (US) 1998-01-15 WO disclosed