SCHEMBL736672

SCHEMBL736672

[Au]C#Cc1ccc(-c2ccccc2)cc1.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
CYP1A1 P04798 1/20 0.48
CYP1B1 Q16678 1/20 0.48
CYP3A4 P08684 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
KCNH2 Q12809 1/20 0.41
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
GRM5 P41594 2/20 0.36
APP P05067 1/20 0.36
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.33
HDAC1 Q13547 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
MAPK1 P28482 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL738589 0.88 CYP3A4 (0.55) CYP1A2CYP3A4TDP1KCNH2ESR1
SCHEMBL738136 0.83 CYP3A4 (0.44) CYP1A2CYP1A1CYP1B1CYP3A4TDP1
SCHEMBL736790 0.79 APP (0.44) CYP3A4TDP1KCNH2APPCA12
SCHEMBL738372 0.78 ALDH1A1 (0.45) CYP3A4TDP1ESR1ESR2GRM5
SCHEMBL739038 0.78 CASP3 (0.49) CYP1A2CYP3A4TDP1ALDH1A1MAPT
SCHEMBL737242 0.76 MAPT (0.44) CYP3A4TDP1GRM5ALDH1A1MAPT
SCHEMBL2018959 0.76 CYP3A4 (0.71) CYP1A2CYP1A1CYP1B1CYP3A4TDP1
SCHEMBL19262009 0.76 CYP3A4 (0.71) CYP1A2CYP1A1CYP1B1CYP3A4TDP1
SCHEMBL30388209 0.76 CYP3A4 (0.71) CYP1A2CYP1A1CYP1B1CYP3A4TDP1
Biphenyl SCHEMBL6633071 0.76 CYP3A4 (0.80) CYP1A2CYP3A4TDP1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847545-B1 SUBSTITUTED ETHYNYL GOLD-NITROGENATED HETEROCYCLIC CARBENE COMPLEX AND ORGANIC ELECTROLUMINESCENT DEVICE USING SAME UBE INDUSTRIES (JP) 2013-03-06 EP disclosed
US-8137821-B2 Substituted ethynyl gold-nitrogen containing heterocyclic carbene complex and organic electroluminescent device using the same UBE INDUSTRIES, LTD. (JP) 2012-03-20 US disclosed
US-20090091243-A1 Substituted Ethynyl Gold-Nitrogen Containing Heterocyclic Carbene Complex and Organic Electroluminescent Device Using the Same UBE INDUSTRIES, LTD. (JP) 2009-04-09 US disclosed
EP-1847545-A1 SUBSTITUTED ETHYNYL GOLD-NITROGENATED HETEROCYCLIC CARBENE COMPLEX AND ORGANIC ELECTROLUMINESCENT DEVICE USING SAME Ube Industries, Ltd. (JP) 2007-10-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090091243-A1 Substituted Ethynyl Gold-Nitrogen Containing Heterocyclic Carbene Complex and Organic Electroluminescent Device Using the Same ACSL3, ATXN2L, ACSL1 CYP1A2 1177/4885CYP1A1 732/4885CYP1B1 1890/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.