SCHEMBL7366940

SCHEMBL7366940

O=C(Oc1ccccc1)n1ncc2ccccc2c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.50
RAB9A P51151 8/20 0.50
PKM P14618 2/20 0.50
MITF O75030 1/20 0.50
PLA2G10 O15496 1/20 0.48
SMN1; SMN2 Q16637 6/20 0.48
ALDH1A1 P00352 4/20 0.48
POLB P06746 1/20 0.48
KDM4E B2RXH2 2/20 0.42
LMNA P02545 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
GLA P06280 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP13 P45452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29462183 0.89 TDP1 (0.44) NPC1RAB9APKMMITFPLA2G10
SCHEMBL7365689 0.81 PLA2G10 (0.55) NPC1RAB9APKMMITFPLA2G10
SCHEMBL10396389 0.80 TFPI2 (0.47) PKMSMN1; SMN2ALDH1A1KDM4EKMT2A
SCHEMBL11310234 0.79 KDM4E (0.46) NPC1RAB9APKMMITFPLA2G10
SCHEMBL21431482 0.78 CYP11B2 (0.44) NPC1RAB9APKMMITFPLA2G10
SCHEMBL31690642 0.78 CYP11B2 (0.44) NPC1RAB9APKMMITFPLA2G10
SCHEMBL9223856 0.77 NPC1 (0.45) NPC1RAB9APKMMITFPLA2G10
SCHEMBL11311967 0.77 PLA2G10 (0.55) NPC1RAB9APKMMITFPLA2G10
SCHEMBL18396652 0.77 RAB9A (0.49) NPC1RAB9APKMMITFSMN1; SMN2
SCHEMBL4580147 0.76 PLA2G10 (0.50) NPC1RAB9APKMMITFPLA2G10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679677-A CARDIOVASCULAR DISORDERS LUITPOLD PHARMA GMBH (DE) 1997-10-21 US disclosed
EP-0649839-A1 Isoquinolinone-, phthalazinone-, quinazolinone- and benzotriazolinone derivatives, their preparation and their use as anti-thrombotics LUITPOLD PHARMA GmbH (DE) 1995-04-26 EP disclosed
WO-1995009842-A1 ISOQUINOLINONE-, PHTHALAZINONE-, QUINAZOLINONE- AND BENZOTRIAZOLINONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ANTI-THROMBOTICS LUITPOLD PHARMA GMBH (DE) 1995-04-13 WO disclosed