SCHEMBL7367335

SCHEMBL7367335

O=C(O)CC1Oc2ccc(C[C@H](NS(=O)(=O)C3CCCCC3)C(=O)OCc3ccccc3)cc2NC1=O

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
HSD17B10 Q99714 3/20 0.39
ALOX15 P16050 2/20 0.39
TSHR P16473 1/20 0.38
USP2 O75604 2/20 0.37
PARP1 P09874 1/20 0.37
IDO1 P14902 1/20 0.36
KMT2A Q03164 1/20 0.36
THRB P10828 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7160888 0.89 TSHR (0.42) GAAHSD17B10TSHRUSP2ALDH1A1
SCHEMBL7368383 0.87 GAA (0.37) GAAHSD17B10ALOX15TSHRKMT2A
SCHEMBL7370120 0.86 HSD17B10 (0.41) GAAHSD17B10ALOX15TSHRUSP2
SCHEMBL7364282 0.86 ALOX15 (0.41) GAAHSD17B10ALOX15USP2PARP1
SCHEMBL7468102 0.86 NPC1 (0.41) GAAHSD17B10TSHRKMT2ATHRB
SCHEMBL7372158 0.85 ITGB3 (0.41) GAAHSD17B10TSHRUSP2KMT2A
SCHEMBL7370705 0.83 HSD17B10 (0.46) GAAHSD17B10ALOX15TSHRUSP2
SCHEMBL7366599 0.83 ITGB3 (0.41) GAAHSD17B10ALOX15USP2PARP1
SCHEMBL7364536 0.82 F10 (0.44) HSD17B10ALOX15
SCHEMBL7589572 0.79 ITGB3 (0.47) HSD17B10TSHRKMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964856-B1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 2002-10-09 EP disclosed
EP-0964856-A1 BICYCLIC AMINO ACIDS MERCK PATENT GmbH (DE) 1999-12-22 EP disclosed
WO-1998035949-A1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 1998-08-20 WO disclosed