SCHEMBL7370705

SCHEMBL7370705

Cc1ccc(S(=O)(=O)N[C@@H](Cc2ccc3c(c2)NC(=O)C(CC(=O)O)O3)C(=O)OCc2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.46
ALOX15 P16050 2/20 0.46
USP2 O75604 1/20 0.45
GAA P10253 1/20 0.45
CTSL P07711 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.44
TSHR P16473 2/20 0.43
HPN P05981 1/20 0.43
ST14 Q9Y5Y6 1/20 0.43
THRB P10828 2/20 0.42
BACE1 P56817 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MMP9 P14780 1/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364282 0.94 ALOX15 (0.41) HSD17B10ALOX15USP2GAACTSL
SCHEMBL7364536 0.90 F10 (0.44) HSD17B10ALOX15HPNST14BACE1
SCHEMBL7163736 0.89 TDP1 (0.53) HSD17B10ALOX15USP2GAASMN1; SMN2
SCHEMBL7365336 0.87 TSHR (0.43) HSD17B10ALOX15SMN1; SMN2TP53POLB
SCHEMBL7370120 0.86 HSD17B10 (0.41) HSD17B10ALOX15USP2GAASMN1; SMN2
SCHEMBL7364374 0.86 ITGB3 (0.44) HSD17B10SMN1; SMN2TP53POLBTSHR
SCHEMBL7165857 0.85 MMP2 (0.47) HSD17B10ALOX15USP2GAAPOLB
SCHEMBL7374002 0.85 SMN1; SMN2 (0.45) HSD17B10ALOX15USP2GAASMN1; SMN2
SCHEMBL7366599 0.84 ITGB3 (0.41) HSD17B10ALOX15USP2GAATHRB
SCHEMBL7367335 0.83 GAA (0.40) HSD17B10ALOX15USP2GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964856-B1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 2002-10-09 EP disclosed
EP-0964856-A1 BICYCLIC AMINO ACIDS MERCK PATENT GmbH (DE) 1999-12-22 EP disclosed
WO-1998035949-A1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 1998-08-20 WO disclosed