SCHEMBL7367467

SCHEMBL7367467

O=C1N(CCC2CCNCC2)CCN1c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.57
DRD3 P35462 5/20 0.53
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
KCNH2 Q12809 4/20 0.45
KHK P50053 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27402876 0.92 DRD2 (0.49) DRD2DRD3MEN1NPC1RAB9A
SCHEMBL11036692 0.86 DRD2 (0.56) DRD2DRD3MEN1NPC1RAB9A
SCHEMBL7392292 0.84 CACNA2D1 (0.46) DRD2DRD3
Hydrochloric Acid SCHEMBL7385931 0.84 CACNA2D1 (0.45) DRD2DRD3
SCHEMBL7394485 0.82 S1PR1 (0.54) DRD2
SCHEMBL7390623 0.82 PRMT1 (0.44) DRD2DRD3
SCHEMBL7390619 0.82 PRMT1 (0.44) DRD2DRD3
Hydrochloric Acid SCHEMBL7393330 0.81 PRMT1 (0.43) DRD2DRD3
Hydrochloric Acid SCHEMBL7395305 0.81 S1PR1 (0.53) DRD2
SCHEMBL7365851 0.81 ACHE (0.62) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997028157-A1 NOVEL PIPERIDINE DERIVATIVES 4-SUBSTITUTED BY AN IMIDAZOLIDIN-2-ON-1-YL-ETHYL, TETRAHYDROPYRIMIDIN-2-ON-1-YL-ETHYL AND 1,3-DIAZEPIN-2-ON-1-YL-ETHYL GROUP, AND USE THEREOF AS α2-ADRENERGIC RECEPTOR ANTAGONISTS PIERRE FABRE MEDICAMENT (FR) 1997-08-07 WO disclosed