SCHEMBL7367480

SCHEMBL7367480

COC(=O)NCN(CCO)c1ccc(C(F)(F)F)cc1C(=O)NCc1ccc(OC)c(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 11/20 0.47
PPARD Q03181 2/20 0.47
PPARG P37231 3/20 0.45
LMNA P02545 2/20 0.45
HPGD P15428 1/20 0.43
GAA P10253 1/20 0.43
TSHR P16473 1/20 0.43
PDE5A O76074 2/20 0.42
PDE6D O43924 1/20 0.42
PDE6A P16499 1/20 0.42
PDE6G P18545 1/20 0.42
PDE6B P35913 1/20 0.42
PDE6C P51160 1/20 0.42
PDE6H Q13956 1/20 0.42
PSEN1 P49768 2/20 0.42
PSEN2 P49810 2/20 0.42
APH1B Q8WW43 2/20 0.42
NCSTN Q92542 2/20 0.42
APH1A Q96BI3 2/20 0.42
PSENEN Q9NZ42 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362850 0.90 PPARA (0.44) PPARAPPARDPPARGLMNAGAA
SCHEMBL7364879 0.90 PPARA (0.47) PPARAPPARDPPARGLMNAGAA
SCHEMBL7361367 0.79 PPARA (0.42) PPARAPPARDPPARGLMNAGAA
SCHEMBL6943273 0.79 PPARA (0.55) PPARAPPARDPPARGLMNAHPGD
SCHEMBL7361602 0.79 PPARA (0.48) PPARAPPARDPPARGLMNAPSEN1
SCHEMBL7372290 0.76 PPARA (0.53) PPARAPPARDPPARGGAAPDE5A
SCHEMBL6941879 0.75 PPARA (0.52) PPARAPPARDPPARGGAAPDE5A
SCHEMBL7391649 0.75 PDE5A (0.46) LMNAHPGDGAAPDE5A
SCHEMBL7372292 0.73 PPARA (0.54) PPARAPPARDPPARGGAAPDE5A
SCHEMBL7368195 0.73 LMNA (0.54) PPARAPPARDPPARGLMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001030745-A1 ANTHRANILIC ACID DERIVATIVES AS INHIBITORS OF THE CGMP-PHOSPHODIESTERASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-03 WO disclosed