SCHEMBL7367595

SCHEMBL7367595

O=C(O)c1ccc(C(=O)c2cccnc2C(=O)O)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.67
ALDH1A1 P00352 3/20 0.67
MAPT P10636 2/20 0.67
CYP3A4 P08684 1/20 0.67
ALOX15 P16050 1/20 0.67
TSHR P16473 1/20 0.67
BLM P54132 1/20 0.67
AGER Q15109 1/20 0.67
NPSR1 Q6W5P4 1/20 0.67
L3MBTL1 Q9Y468 1/20 0.67
TDP1 Q9NUW8 1/20 0.48
SRD5A2 P31213 2/20 0.48
DHODH Q02127 1/20 0.48
CYP2C8 P10632 1/20 0.47
CYP2C9 P11712 1/20 0.47
GAA P10253 1/20 0.47
CYP1A2 P05177 1/20 0.46
NAPRT Q6XQN6 2/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL296670 0.91 KDM4E (0.69) KDM4EALDH1A1MAPTCYP3A4ALOX15
Hydrochloric Acid SCHEMBL7853761 0.89 KDM4E (0.67) KDM4EALDH1A1MAPTCYP3A4ALOX15
Terephthalic Acid SCHEMBL28292423 0.89 KDM4E (0.85) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL6987666 0.88 ALDH1A1 (0.61) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL7529815 0.88 KDM4E (0.61) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL2212405 0.88 KDM4E (0.61) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL7364079 0.88 KDM4E (0.61) KDM4EALDH1A1MAPTCYP3A4ALOX15
Oxalic Acid SCHEMBL31550428 0.88 KDM4E (0.65) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL9635664 0.87 KDM4E (0.80) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL7369102 0.86 KDM4E (0.67) KDM4EALDH1A1MAPTCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652218-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-07-11 EP disclosed
CN-1052004-C Heterocyclic compounds, their production and use TALCEDA CHEMICAL IND LTD (JP) 2000-05-03 CN disclosed
US-5716954-A ANTIINFLAMMATORY AGENT, ANTIHISTAMINES, IMMUNOSUPPRESSION,AUTOIMMUNE DISEASES SYNTEX U.S.A. INC. (US) 1998-02-10 US disclosed
US-5585385-A USEFUL IN TREATING DISORDERS OF MICTURITION; ADMINISTERING TO INHIBIT PLASMA EXTRAVASATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-17 US disclosed
CN-1107476-A Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-08-30 CN disclosed
EP-0652218-A1 Heterocyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-05-10 EP disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed
US-4259527-A OXIDATION OF SECONDARY ALCOHOLS TO KETONES WITH HYDROGEN PEROXIDE ALLIED CHEMICAL CORPORATION (US) 1981-03-31 US disclosed
US-4171313-A OF ALICYCLIC KETONES TO LACTONES, W-HYDROXY ACIDS AND ESTERS USING HYDROGEN PEROXIDE AS AN OXIDIZING AGENT ALLIED CHEMICAL CORPORATION (US) 1979-10-16 US disclosed