SCHEMBL7367635

SCHEMBL7367635

Cc1cccc2[nH]nc(C(=O)OC3CC4CCC(C3)N4C)c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 3/20 0.52
HTR3B O95264 3/20 0.52
HTR3A P46098 3/20 0.52
HTR3D Q70Z44 3/20 0.52
HTR3C Q8WXA8 3/20 0.52
CHRNA7 P36544 2/20 0.52
CYP2D6 P10635 2/20 0.50
CHRNA1 P02708 1/20 0.50
CHRNG P07510 1/20 0.50
CYP3A4 P08684 1/20 0.50
HTR1A P08908 1/20 0.50
CHRM5 P08912 1/20 0.50
MAPT P10636 1/20 0.50
CHRM1 P11229 1/20 0.50
CHRNB1 P11230 1/20 0.50
CHRNB2 P17787 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
CHRM3 P20309 1/20 0.50
CHRNB4 P30926 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23153182 0.84 HTR3A (0.53) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9876004 0.82 GSK3B (0.55) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL3779528 0.72 MAP2K4 (0.49) MAPTSMN1; SMN2
SCHEMBL22725235 0.70 HTR3A (0.71) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7652481 0.70 HTR3A (0.75) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7652475 0.70 HTR3A (0.75) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL570533 0.70 HAO1 (0.50) MAPTSMN1; SMN2
SCHEMBL6507484 0.69 HTR3E (0.72) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL6507481 0.69 HTR3E (0.72) HTR3EHTR3BHTR3AHTR3DHTR3C
Benzoyl Tropine SCHEMBL221830 0.69 HTR3E (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0200444-A2 Azabicyclononyl-indazole-carboxamide having 5-HT antagonist activity BEECHAM GROUP PLC (GB) 1986-11-05 EP claimed