SCHEMBL7368769

SCHEMBL7368769

CSc1sc(-c2ncco2)c2c1CCCC2

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.34
ELANE P08246 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7463979 0.81 LRRK2 (0.57) LRRK2
SCHEMBL23629116 0.60
SCHEMBL100765 0.60 HPGDS (0.46)
SCHEMBL24912726 0.57 LTA4H (0.50)
SCHEMBL3026407 0.55
SCHEMBL3901936 0.54 MAPK8 (0.40)
SCHEMBL21852154 0.54 NOS3 (0.36)
SCHEMBL28459432 0.54 HPGDS (0.33)
SCHEMBL23254437 0.53 HPGDS (0.46) LRRK2
SCHEMBL24156800 0.53 ATM (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001503408-A 2001-03-13 JP claimed
EP-0937072-A1 THIENYLCYCLOHEXANONE DERIVATIVES AS LIGANDS OF THE GABA A? $g(a)5 RECEPTOR SUBTYPE MERCK SHARP & DOHME LTD. (GB) 1999-08-25 EP claimed
WO-1998018792-A1 THIENYLCYCLOHEXANONE DERIVATIVES AS LIGANDS OF THE GABAA α5 RECEPTOR SUBTYPE MERCK SHARP & DOHME LIMITED (GB) 1998-05-07 WO claimed