SCHEMBL7369543

SCHEMBL7369543

O=C(O)CCCCCCc1cc(-c2nc3ccccc3[nH]c2=O)cc([N+](=O)[O-])c1CCCCCCC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.44
RAB9A P51151 4/20 0.44
NPC1 O15118 3/20 0.44
MAPT P10636 2/20 0.39
DAGLA Q9Y4D2 1/20 0.39
CHRM1 P11229 1/20 0.39
FBP1 P09467 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HSD17B10 Q99714 2/20 0.37
HPGD P15428 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
PKM P14618 2/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
SERPINE1 P05121 1/20 0.37
MAPK1 P28482 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364700 0.78 MMP2 (0.48) KDM4ERAB9ANPC1MAPTCHRM1
SCHEMBL7364869 0.77 PRKAG1 (0.47) RAB9ANPC1MAPTFBP1LMNA
SCHEMBL7366603 0.73 NPC1 (0.53) KDM4ERAB9ANPC1MAPTALDH1A1
SCHEMBL8726193 0.72 KDM4E (0.42) KDM4ERAB9ANPC1MAPTDAGLA
SCHEMBL8726189 0.69 MAPT (0.53) KDM4ERAB9ANPC1MAPTFBP1
SCHEMBL7371644 0.69 ALDH1A1 (0.47) FBP1ALDH1A1
SCHEMBL7367829 0.69 MAPT (0.53) KDM4ERAB9ANPC1MAPTFBP1
SCHEMBL7375356 0.69 RAB9A (0.45) KDM4ERAB9ANPC1MAPTALDH1A1
SCHEMBL6754408 0.68 MAPT (0.54) RAB9ANPC1MAPTALDH1A1HPGD
SCHEMBL4610015 0.68 MAPT (0.54) RAB9ANPC1MAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237929-B1 3,5-DISUBSTITUTED PYROCATECHOL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-06-02 EP disclosed
EP-0237929-A1 3,5-Disubstituted pyrocatechol derivatives F. HOFFMANN-LA ROCHE AG (CH) 1987-09-23 EP disclosed