SCHEMBL736956

SCHEMBL736956

COc1ccc2[nH]cc(C)c2c1.COc1ccc2[nH]cc(C)c2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 2/20 0.64
HTR2B P41595 5/20 0.60
CYP1A2 P05177 3/20 0.60
ALDH1A1 P00352 2/20 0.60
CYP2C19 P33261 1/20 0.60
HTR2A P28223 6/20 0.57
HTR2C P28335 5/20 0.57
MAPT P10636 3/20 0.57
HTR1A P08908 3/20 0.57
TSHR P16473 2/20 0.57
CYP2D6 P10635 2/20 0.57
HTR1D P28221 2/20 0.57
HTR1B P28222 2/20 0.57
HTR7 P34969 2/20 0.57
HTR6 P50406 2/20 0.57
HTR4 Q13639 2/20 0.57
NFKB1 P19838 1/20 0.57
TRPM8 Q7Z2W7 1/20 0.57
NR4A2 P43354 1/20 0.57
KDM4E B2RXH2 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL434877 1.00 GPR84 (0.64) GPR84HTR2BCYP1A2ALDH1A1CYP2C19
SCHEMBL1120777 0.85 KDM4E (0.60) GPR84HTR2BCYP1A2ALDH1A1CYP2C19
SCHEMBL5432612 0.82 GPR84 (0.66) GPR84HTR2BCYP1A2ALDH1A1CYP2C19
SCHEMBL3629976 0.81 HTR2B (0.65) GPR84HTR2BCYP1A2ALDH1A1CYP2C19
SCHEMBL28337310 0.81 GPR84 (0.64) GPR84HTR2BCYP1A2ALDH1A1CYP2C19
SCHEMBL23259474 0.80 HTR1B (0.52) GPR84HTR2BCYP1A2CYP2C19HTR2A
SCHEMBL6290566 0.79 GPR84 (0.62) GPR84HTR2BCYP1A2ALDH1A1CYP2C19
SCHEMBL21256024 0.79 GPR84 (0.62) GPR84HTR2BCYP1A2ALDH1A1CYP2C19
SCHEMBL21623872 0.79 GPR84 (0.62) GPR84HTR2BCYP1A2ALDH1A1CYP2C19
SCHEMBL4475932 0.79 GPR84 (0.62) GPR84HTR2BCYP1A2ALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138187-B2 Substituted heteroaryl derivatives GRUENENTHAL GMBH (DE) 2012-03-20 US disclosed