SCHEMBL7370205

SCHEMBL7370205

COc1ccc(CN)cc1OCC(=O)N1CCN(Cc2ccc(Cl)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.56
KDM4E B2RXH2 5/20 0.55
MAPK1 P28482 2/20 0.55
MEN1 O00255 1/20 0.55
TP53 P04637 1/20 0.55
KMT2A Q03164 1/20 0.55
CYP3A4 P08684 3/20 0.54
ALDH1A1 P00352 3/20 0.54
CYP2C9 P11712 1/20 0.54
LMNA P02545 3/20 0.53
DRD3 P35462 2/20 0.53
ABCB11 O95342 1/20 0.53
CYP1A2 P05177 1/20 0.53
ADRA2A P08913 1/20 0.53
CYP2D6 P10635 1/20 0.53
CHRM1 P11229 1/20 0.53
TBXA2R P21731 1/20 0.53
SLC6A2 P23975 1/20 0.53
SLC6A4 P31645 1/20 0.53
CYP2C19 P33261 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5063868 0.96 CCR1 (0.56) CCR1KDM4EMAPK1MEN1TP53
SCHEMBL7370428 0.92 ALDH1A1 (0.62) KDM4EMAPK1MEN1TP53KMT2A
SCHEMBL7369950 0.92 KDM4E (0.55) CCR1KDM4EMAPK1MEN1TP53
SCHEMBL5064235 0.91 CCR1 (0.58) CCR1KDM4EMAPK1MEN1TP53
SCHEMBL8545193 0.91 KDM4E (0.54) KDM4EMAPK1MEN1TP53KMT2A
SCHEMBL5061535 0.89 CCR1 (0.56) CCR1KDM4EMAPK1MEN1TP53
SCHEMBL5064434 0.88 KDM4E (0.58) CCR1KDM4EMAPK1MEN1TP53
SCHEMBL5064511 0.88 CCR1 (0.55) CCR1KDM4EMAPK1MEN1TP53
SCHEMBL5066421 0.87 CCR1 (0.58) CCR1KDM4EMAPK1MEN1TP53
SCHEMBL5060462 0.87 CCR1 (0.63) CCR1KDM4EMAPK1MEN1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706517-B1 PYRIDAZINONE DERIVATIVES WITH PHARMACEUTICAL ACTIVITY NISSAN CHEMICAL IND LTD (JP) 1998-10-21 EP disclosed
EP-0706517-A1 PYRIDAZINONE DERIVATIVES WITH PHARMACEUTICAL ACTIVITY NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1996-04-17 EP disclosed
WO-1995001343-A1 PYRIDAZINONE DERIVATIVES WITH PHARMACEUTICAL ACTIVITY NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1995-01-12 WO disclosed