SCHEMBL7370356

SCHEMBL7370356

CCOC(=O)c1ccccc1N(C)C(=O)c1ccc(N)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
HSD17B10 Q99714 1/20 0.48
HSD17B2 P37059 1/20 0.44
TSHR P16473 2/20 0.43
MAPT P10636 3/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 2/20 0.42
HTT P42858 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CDC25B P30305 3/20 0.41
SIRT3 Q9NTG7 1/20 0.40
HTR4 Q13639 1/20 0.40
ERN1 O75460 1/20 0.40
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374190 0.83 ALDH1A1 (0.48) ALDH1A1HSD17B2TSHRMAPTKDM4E
SCHEMBL7378235 0.82 GPBAR1 (0.45) ALDH1A1HSD17B2TSHRHTTSMN1; SMN2
SCHEMBL7374024 0.82 LMNA (0.55) ALDH1A1HSD17B10TSHRMAPTKDM4E
SCHEMBL7368763 0.82 RAB9A (0.43) ALDH1A1TSHRMAPTHPGDGAA
SCHEMBL7376664 0.81 CYP1A2 (0.45) ALDH1A1HSD17B10TSHRMAPTGAA
SCHEMBL1612538 0.78 HSD17B2 (0.69) HSD17B2TSHRMAPTKDM4EGAA
SCHEMBL7341812 0.77 RAB9A (0.39) ALDH1A1TSHRMAPTKDM4ERAB9A
SCHEMBL7373084 0.76 ALDH1A1 (0.47) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL7376544 0.76 ALDH1A1 (0.49) ALDH1A1TSHRMAPTKDM4EGAA
SCHEMBL7371851 0.74 CYP1A2 (0.43) ALDH1A1HSD17B10HSD17B2TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed