SCHEMBL7378235

SCHEMBL7378235

COc1cc(C(=O)N(C)c2ccccc2C)ccc1N

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.45
HSD17B1 P14061 8/20 0.43
HSD17B2 P37059 7/20 0.43
STS P08842 5/20 0.43
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HSD11B1 P28845 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7376664 0.88 CYP1A2 (0.45) GPBAR1TSHRSMN1; SMN2MEN1KMT2A
SCHEMBL7373607 0.85 HSD17B1 (0.44) GPBAR1HSD17B1HSD17B2TSHRSMN1; SMN2
SCHEMBL7370356 0.82 ALDH1A1 (0.48) HSD17B2TSHRSMN1; SMN2MEN1KMT2A
SCHEMBL7371851 0.81 CYP1A2 (0.43) HSD17B1HSD17B2TSHRMEN1KMT2A
SCHEMBL7371278 0.80 ALDH1A1 (0.44) GPBAR1TSHRSMN1; SMN2MEN1KMT2A
SCHEMBL7368763 0.80 RAB9A (0.43) TSHRSMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL7968869 0.79 KMT2A (0.49) SMN1; SMN2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL358787 0.78 ALDH1A1 (0.50) TSHRSMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL7425044 0.78 DRD2 (0.46) SMN1; SMN2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL7422014 0.77 SMN1; SMN2 (0.47) TSHRSMN1; SMN2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed