SCHEMBL7370446

SCHEMBL7370446

COC(=O)C[C@H]1C(=O)N(OC(=O)COC(=O)C(F)(F)F)CCN1C(=O)C(C)NC(=O)c1ccc(-c2ccncc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PREP P48147 1/20 0.38
FAP Q12884 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
ROCK2 O75116 12/20 0.34
ROCK1 Q13464 8/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
ITGB3 P05106 4/20 0.33
ITGA2B P08514 4/20 0.33
PRKG1 Q13976 3/20 0.33
RPS6KA5 O75582 2/20 0.33
CDK1 P06493 2/20 0.33
PRKACA P17612 2/20 0.33
RPS6KB1 P23443 2/20 0.33
CDK2 P24941 2/20 0.33
MAPK1 P28482 2/20 0.33
GSK3A P49840 2/20 0.33
GSK3B P49841 2/20 0.33
PRKX P51817 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366992 0.84 ALDH1A1 (0.34) ALDH1A1MAPTITGB3ITGA2BLMNA
SCHEMBL7931569 0.84 ITGB3 (0.42) PREPFAPDPP8DPP9ROCK2
Trifluoroacetic Acid SCHEMBL7370443 0.81 ITGB3 (0.49) PREPFAPDPP8DPP9ROCK2
Trifluoroacetic Acid SCHEMBL7931567 0.81 ITGB3 (0.49) PREPFAPDPP8DPP9ROCK2
SCHEMBL7372733 0.78 ITGB3 (0.43) PREPFAPDPP8DPP9ROCK2
SCHEMBL7372729 0.78 ITGB3 (0.43) PREPFAPDPP8DPP9ROCK2
SCHEMBL7372732 0.78 ITGB3 (0.43) PREPFAPDPP8DPP9ROCK2
SCHEMBL7364293 0.76 DPP8 (0.41) FAPDPP8ROCK2ALDH1A1ITGB3
SCHEMBL7374179 0.72 ITGB3 (0.40) ROCK2ROCK1ITGB3ITGA2BPRKG1
Trifluoroacetic Acid SCHEMBL7931550 0.70 ITGB3 (0.48) ROCK2ROCK1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed