SCHEMBL7366992

SCHEMBL7366992

COC(=O)C[C@H]1C(=O)N(OC(=O)COC(=O)C(F)(F)F)CCN1C(=O)C(C)NC(=O)c1ccc(C2CCNCC2)cc1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
ITGB3 P05106 9/20 0.34
ITGA2B P08514 9/20 0.34
CCR1 P32246 5/20 0.34
SYK P43405 2/20 0.34
ITGA2 P17301 2/20 0.34
LMNA P02545 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7924872 0.85 ITGB3 (0.40) ALDH1A1MAPTITGB3ITGA2BCCR1
SCHEMBL7370446 0.84 PREP (0.38) ALDH1A1MAPTITGB3ITGA2BLMNA
Trifluoroacetic Acid SCHEMBL7366990 0.82 ITGB3 (0.48) ITGB3ITGA2BCCR1ITGA2LMNA
SCHEMBL7924876 0.68 ITGB3 (0.49) ITGB3ITGA2BITGA2KMT2A
SCHEMBL7924873 0.68 ITGB3 (0.49) ITGB3ITGA2BITGA2KMT2A
SCHEMBL7364293 0.67 DPP8 (0.41) ALDH1A1ITGB3ITGA2B
Trifluoroacetic Acid SCHEMBL7931567 0.66 ITGB3 (0.49) ITGB3ITGA2B
Trifluoroacetic Acid SCHEMBL7370443 0.66 ITGB3 (0.49) ITGB3ITGA2B
SCHEMBL7372732 0.63 ITGB3 (0.43) ITGB3ITGA2BKMT2A
SCHEMBL7372733 0.63 ITGB3 (0.43) ITGB3ITGA2BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed