SCHEMBL7370587

SCHEMBL7370587

[CH2]c1cccc(C(=O)Nn2ncc(C)n2)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
LMNA P02545 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
GRM5 P41594 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP3A4 P08684 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
THRB P10828 1/20 0.34
GAA P10253 1/20 0.34
CYP2D6 P10635 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374400 0.84 ADORA2A (0.37) ALDH1A1LMNANPC1RAB9AHDAC8
SCHEMBL7378561 0.84 LMNA (0.34) ALDH1A1LMNAHDAC8HDAC6CYP2C9
SCHEMBL7379897 0.83 LMNA (0.34) ALDH1A1LMNANPC1RAB9AHDAC8
SCHEMBL7379117 0.83 LMNA (0.34) ALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL7376359 0.81 ADORA2A (0.35) ALDH1A1LMNANPC1RAB9AHDAC8
SCHEMBL7376717 0.80 MAPT (0.35) ALDH1A1LMNAGRM5CYP2C19SMN1; SMN2
SCHEMBL7375838 0.80 LMNA (0.38) ALDH1A1LMNANPC1HDAC8HDAC6
SCHEMBL1196695 0.69 HDAC8 (0.63) ALDH1A1HDAC8HDAC6SMN1; SMN2THRB
SCHEMBL7698185 0.68 HTT (0.58) LMNANPC1RAB9AHDAC8HDAC6
SCHEMBL7698519 0.68 HTT (0.63) LMNANPC1RAB9AHDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO claimed
US-5763469-A Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-06-09 US disclosed
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO disclosed