SCHEMBL7376359

SCHEMBL7376359

[CH2]c1cccc(C(=O)Nn2ncc(NCC)n2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
HCAR3 P49019 1/20 0.35
ALDH1A1 P00352 2/20 0.33
FYN P06241 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
DYRK1A Q13627 4/20 0.32
DYRK2 Q92630 4/20 0.32
DYRK1B Q9Y463 4/20 0.32
DYRK3 O43781 3/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
LCK P06239 1/20 0.32
BTK Q06187 1/20 0.32
CDK8 P49336 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374400 0.86 ADORA2A (0.37) ADORA2AADORA1ALDH1A1FYNLMNA
SCHEMBL7379117 0.83 LMNA (0.34) ALDH1A1LMNASMN1; SMN2
SCHEMBL7370587 0.81 ALDH1A1 (0.37) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL7376717 0.80 MAPT (0.35) ALDH1A1LMNASMN1; SMN2
SCHEMBL7378561 0.79 LMNA (0.34) ADORA2AADORA1ALDH1A1LMNAPOLB
SCHEMBL7379897 0.78 LMNA (0.34) ADORA2AADORA1ALDH1A1LMNASMN1; SMN2
SCHEMBL7375838 0.75 LMNA (0.38) ALDH1A1LMNANPC1HDAC8HDAC6
SCHEMBL7381168 0.70 ADORA2A (0.37) ADORA2AADORA1
SCHEMBL1197188 0.70 SMN1; SMN2 (0.53) ALDH1A1SMN1; SMN2NPC1RAB9ACDK8
SCHEMBL7375884 0.70 MEN1 (0.39) ALDH1A1LMNASMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO claimed
US-5763469-A Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-06-09 US disclosed
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO disclosed