SCHEMBL7378561

SCHEMBL7378561

[CH2]c1cccc(C(=O)Nn2ncc(N)n2)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.34
PTGS1 P23219 2/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 1/20 0.33
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
AOC2 O75106 1/20 0.32
FURIN P09958 1/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KLKB1 P03952 2/20 0.31
MEN1 O00255 2/20 0.31
MAPT P10636 2/20 0.31
KMT2A Q03164 2/20 0.31
KDM1A O60341 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7370587 0.84 ALDH1A1 (0.37) LMNAALDH1A1KDM4EHDAC8HDAC6
SCHEMBL7374400 0.82 ADORA2A (0.37) LMNAALDH1A1HDAC8HDAC6CYP2D6
SCHEMBL7379117 0.81 LMNA (0.34) LMNAALDH1A1KDM4E
SCHEMBL7379897 0.81 LMNA (0.34) LMNAALDH1A1KDM4EHDAC8HDAC6
SCHEMBL7375838 0.80 LMNA (0.38) LMNAALDH1A1KDM4EHDAC8HDAC6
SCHEMBL7376359 0.79 ADORA2A (0.35) LMNAALDH1A1HDAC8HDAC6POLB
SCHEMBL7376717 0.78 MAPT (0.35) LMNAALDH1A1PKMCYP2C19MEN1
SCHEMBL7698185 0.68 HTT (0.58) LMNAHDAC8HDAC6POLBCYP2D6
SCHEMBL7698519 0.68 HTT (0.63) LMNAHDAC8HDAC6POLBCYP2D6
SCHEMBL7376224 0.67 MEN1 (0.33) LMNAPTGS1ALDH1A1KDM4EHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO claimed
US-5763469-A Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-06-09 US disclosed
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO disclosed