SCHEMBL7370662

SCHEMBL7370662

CC(C)(C)OC(=O)CN1CCC(C(=O)Nc2ccc(N3CCNCC3)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN2 P17706 1/20 0.51
PTPN1 P18031 1/20 0.51
PTPN6 P29350 1/20 0.51
WNT1 P04628 1/20 0.47
GSK3B P49841 1/20 0.47
DYRK1A Q13627 1/20 0.47
ABL1 P00519 2/20 0.45
RIN1 Q13671 1/20 0.45
MAPK1 P28482 3/20 0.45
ALDH1A1 P00352 2/20 0.45
ME3 Q16798 1/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
RAD52 P43351 1/20 0.42
GFER P55789 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8143555 0.89 ALDH1A1 (0.48) WNT1GSK3BDYRK1AABL1MAPK1
SCHEMBL8140931 0.89 PTPN2 (0.52) PTPN2PTPN1PTPN6WNT1GSK3B
SCHEMBL8135054 0.87 LMNA (0.49) ABL1MAPK1ALDH1A1ME3RAB9A
SCHEMBL7376347 0.84 ALDH1A1 (0.43) ABL1MAPK1ALDH1A1ME3MEN1
SCHEMBL7371765 0.84 ME3 (0.54) ABL1MAPK1ALDH1A1ME3MEN1
SCHEMBL7375251 0.83 PTPN2 (0.61) PTPN2PTPN1PTPN6ABL1RIN1
Trifluoroacetic Acid SCHEMBL7376343 0.80 ME3 (0.48) ABL1MAPK1ALDH1A1ME3MEN1
Acetic Acid SCHEMBL8135057 0.80 ME3 (0.52) ABL1MAPK1ALDH1A1ME3NPC1
Acetic Acid SCHEMBL7375335 0.80 ME3 (0.52) PTPN2PTPN1PTPN6ABL1ALDH1A1
SCHEMBL8144011 0.80 PTPN2 (0.62) PTPN2PTPN1PTPN6ABL1RIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140792-A1 3,4-DIAMINO-3-CYCLOBUTENE-1,2-DIONE DERIVATIVES WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-10 EP claimed
WO-2000035855-A1 3,4-DIAMINO-3-CYCLOBUTENE-1,2-DIONE DERIVATIVES WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-22 WO claimed