SCHEMBL7375263

SCHEMBL7375263

Cc1ccc(N(C)C(=O)c2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.56
HSD17B10 Q99714 1/20 0.56
ATM Q13315 1/20 0.56
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
ALDH1A1 P00352 3/20 0.50
PKM P14618 1/20 0.50
MAPK1 P28482 1/20 0.50
CES1 P23141 1/20 0.49
CRHBP P24387 2/20 0.48
CRHR2 Q13324 2/20 0.48
MEN1 O00255 1/20 0.48
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31155755 0.89 ATM (0.57) ATMALDH1A1MAPK1CES1CRHBP
SCHEMBL20474766 0.86 ATM (0.55) ACHEHSD17B10ATMALDH1A1MAPK1
SCHEMBL7376913 0.86 ATM (0.55) ATMMAOAMAOBALDH1A1MAPK1
SCHEMBL7379932 0.86 ATM (0.75) ATMMAOAALDH1A1MAPK1CES1
SCHEMBL12938525 0.85 HSD17B1 (0.57) MAOAALDH1A1CES1KMT2ASMN1; SMN2
SCHEMBL7375652 0.84 ALDH1A1 (0.55) ATMMAOAMAOBALDH1A1MAPK1
SCHEMBL15480653 0.84 ATM (0.52) ATMALDH1A1MAPK1MEN1POLB
SCHEMBL7376372 0.82 HSD17B1 (0.64) ACHEATMALDH1A1MAPK1CRHBP
SCHEMBL18585670 0.80 ALDH1A1 (0.51) ACHEHSD17B10ATMALDH1A1MAPK1
SCHEMBL25491787 0.80 HSD17B1 (0.59) ALDH1A1POLBKMT2ASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed