SCHEMBL7375589

SCHEMBL7375589

Oc1ccc2o[c]nc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.42
ESR1 P03372 12/20 0.42
ESR2 Q92731 12/20 0.42
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 1/20 0.38
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
KMT2A Q03164 1/20 0.34
CA12 O43570 2/20 0.33
CA9 Q16790 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4152683 0.75 RAB9A (0.42) PIK3CBALDH1A1KDM4EHPGDLMNA
SCHEMBL938963 0.75 NPC1 (0.42) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL207390 0.75 LMNA (0.44) ALDH1A1KDM4EHPGDLMNAMAPT
SCHEMBL207265 0.75 AHR (0.37) PIK3CAALDH1A1MAPTALOX15HTT
SCHEMBL7288719 0.75 CA12 (0.39) ALDH1A1HSD17B10MEN1KMT2ACA12
SCHEMBL940594 0.72 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDLMNAMAPT
SCHEMBL3572976 0.72 RAB9A (0.47) ALDH1A1HPGDMAPTSMN1; SMN2MEN1
SCHEMBL5337212 0.71 CYP2A6 (0.42) ALDH1A1KDM4E
SCHEMBL11784689 0.71 RAB9A (0.42) ALDH1A1KDM4EHPGDMAPTALOX15
SCHEMBL407727 0.71 PKM (0.45) KDM4ESMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164371-A HETEROCYCLIC KETONES ICI AMERICAS INC. (US) 1992-11-17 US disclosed
EP-0291234-A2 Peptidic human leukocyte elastase (HLE) inhibitors ZENECA INC. (US) 1988-11-17 EP disclosed