SCHEMBL7375760

SCHEMBL7375760

CCOC(=O)CCc1ccc(CCNC(=O)c2cccc(C#N)c2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.67
RAB9A P51151 6/20 0.49
NPC1 O15118 5/20 0.49
ROCK2 O75116 1/20 0.48
EPHX2 P34913 2/20 0.46
ALOX5 P09917 1/20 0.46
CYP4F2 P78329 1/20 0.46
CYP4A11 Q02928 1/20 0.46
NAMPT P43490 1/20 0.45
MAPT P10636 3/20 0.45
HDAC3 O15379 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458374 0.91 GAA (0.56) GAAROCK2EPHX2CYP4F2CYP4A11
SCHEMBL7864682 0.86 GAA (0.55) GAARAB9AROCK2EPHX2ALOX5
SCHEMBL6881434 0.80 FFAR1 (0.52) GAACYP4F2CYP4A11POLB
SCHEMBL12988864 0.77 L3MBTL1 (0.63) GAARAB9ANPC1ROCK2NAMPT
SCHEMBL4506493 0.77 CYP4F2 (0.66) RAB9ACYP4F2CYP4A11MAPT
SCHEMBL9267010 0.76 RAB9A (0.62) GAARAB9ANPC1EPHX2MAPT
SCHEMBL3984665 0.76 GAA (0.64) GAARAB9ANPC1ROCK2NAMPT
SCHEMBL6359399 0.75 SMN1; SMN2 (0.72) GAANAMPTMAPTHDAC3SMN1; SMN2
SCHEMBL1659817 0.75 GSK3B (0.57) GAASMN1; SMN2GPR139GRM5MEN1
SCHEMBL8497478 0.74 LMNA (0.53) GAARAB9ANPC1MAPTHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP disclosed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed