SCHEMBL7864682

SCHEMBL7864682

CCOC(=O)CCc1cccc(CNC(=O)c2cccc(C#N)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.55
CHRM3 P20309 2/20 0.50
ROCK2 O75116 6/20 0.46
ROCK1 Q13464 1/20 0.46
PPARG P37231 1/20 0.46
MMP13 P45452 1/20 0.46
EPHX2 P34913 2/20 0.45
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
ADORA2A P29274 1/20 0.44
RAB9A P51151 1/20 0.43
MAOA P21397 1/20 0.43
GPR139 Q6DWJ6 1/20 0.43
VNN1 O95497 1/20 0.43
GRM5 P41594 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
ALOX5 P09917 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458374 0.93 GAA (0.56) GAACHRM3ROCK2ROCK1PPARG
SCHEMBL7375760 0.86 GAA (0.67) GAAROCK2EPHX2RAB9AGPR139
SCHEMBL6881434 0.84 FFAR1 (0.52) GAAPPARG
SCHEMBL7380693 0.82 F10 (0.51) ROCK2PPARGMMP13EPHX2LMNA
SCHEMBL7862007 0.80 MMP13 (0.47) ROCK2ROCK1PPARGMMP13EPHX2
SCHEMBL7861961 0.80 SENP1 (0.49) ROCK2PPARGMMP13EPHX2LMNA
SCHEMBL7862004 0.80 MMP13 (0.47) ROCK2ROCK1PPARGMMP13EPHX2
SCHEMBL7380699 0.79 PPARG (0.44) GAAROCK2PPARGMMP13EPHX2
SCHEMBL7862050 0.79 PPARG (0.44) ROCK2PPARGMMP13EPHX2LMNA
SCHEMBL7861953 0.78 NAMPT (0.55) PPARGLMNAHPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed