SCHEMBL7375795

SCHEMBL7375795

CN(C)CCOc1cccc(-c2cc(=O)c3c(O)cc(O)cc3o2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLH Q9Y253 2/20 0.61
QPCT Q16769 2/20 0.60
ABCB1 P08183 2/20 0.59
XDH P47989 6/20 0.57
CYP1A1 P04798 3/20 0.57
CYP1A2 P05177 3/20 0.57
HDAC8 Q9BY41 2/20 0.57
HDAC6 Q9UBN7 2/20 0.57
MEN1 O00255 2/20 0.57
ALDH1A1 P00352 2/20 0.57
TP53 P04637 2/20 0.57
CYP3A4 P08684 2/20 0.57
CYP2D6 P10635 2/20 0.57
MAPT P10636 2/20 0.57
CYP2C9 P11712 2/20 0.57
MAOA P21397 2/20 0.57
MAOB P27338 2/20 0.57
MAPK1 P28482 2/20 0.57
CYP2C19 P33261 2/20 0.57
KMT2A Q03164 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10433113 0.82 SIGMAR1 (0.59) CYP1A1CYP1A2MAOBSIGMAR1CYP2B6
SCHEMBL433900 0.82 EGFR (0.71) ABCB1CYP1A1CYP1A2CYP3A4MAPT
SCHEMBL16823312 0.81 EGFR (0.70) ABCB1MAPTSIGMAR1EGFRRET
SCHEMBL431393 0.80 EGFR (0.69) SIGMAR1EGFRRETKDR
SCHEMBL4152555 0.77 ABCB1 (0.93) POLHQPCTABCB1XDHCYP1A1
SCHEMBL31291006 0.77 POLH (1.00) POLHQPCTABCB1XDHCYP1A1
SCHEMBL30335147 0.77 POLH (1.00) POLHQPCTABCB1XDHCYP1A1
Chrysin SCHEMBL28168227 0.75 MAPT (0.89) POLHQPCTABCB1XDHCYP1A1
SCHEMBL4152249 0.74 ABCB1 (1.00) POLHQPCTABCB1XDHCYP1A1
SCHEMBL4156163 0.74 ABCB1 (1.00) POLHQPCTABCB1XDHCYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115718-A1 HYDROXYFLAVONE DERIVATIVES AS TAU PROTEIN KINASE 1 INHIBITORS MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000017184-A1 HYDROXYFLAVONE DERIVATIVES AS TAU PROTEIN KINASE 1 INHIBITORS MITSUBISHI CHEMICAL CORPORATION (JP) 2000-03-30 WO disclosed