SCHEMBL7375896

SCHEMBL7375896

CCOC(=O)CN(C(=O)c1ccc([N+](=O)[O-])cc1)c1ccccc1C

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
NPSR1 Q6W5P4 1/20 0.46
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
KMT2A Q03164 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 2/20 0.42
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
TSHR P16473 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957845 0.90 ALDH1A1 (0.50) ALDH1A1CRHBPCRHR2LMNAMAPT
SCHEMBL7419641 0.86 ALDH1A1 (0.52) ALDH1A1CRHBPCRHR2LMNAMAPT
SCHEMBL7417406 0.83 ALDH1A1 (0.70) ALDH1A1CRHBPCRHR2LMNAMAPT
SCHEMBL7367843 0.83 NPSR1 (0.49) ALDH1A1NPSR1LMNAMAPTKDM4E
SCHEMBL7372075 0.80 CRHBP (0.65) ALDH1A1NPSR1CRHBPCRHR2LMNA
SCHEMBL7422213 0.79 ALDH1A1 (0.54) ALDH1A1CRHBPCRHR2LMNAMAPT
SCHEMBL3453497 0.78 CRHBP (0.70) ALDH1A1CRHBPCRHR2LMNAMAPT
SCHEMBL7416266 0.77 ALDH1A1 (0.54) ALDH1A1LMNAMAPTKDM4EKMT2A
SCHEMBL8103391 0.76 ALDH1A1 (0.53) ALDH1A1MAPTKDM4EKMT2AMEN1
SCHEMBL7371730 0.76 CRHBP (0.51) ALDH1A1CRHBPCRHR2MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed