SCHEMBL7377115

SCHEMBL7377115

COc1scc(C)c1-c1nc(-c2cccnc2)c(C)[nH]1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 6/20 0.57
CYP2A6 P11509 4/20 0.40
CYP2E1 P05181 3/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2C9 P11712 3/20 0.40
CYP2B6 P20813 3/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 2/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP19A1 P11511 4/20 0.39
SMPD3 Q9NY59 1/20 0.39
HPGDS O60760 1/20 0.37
KIT P10721 1/20 0.37
CYP11B1 P15538 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7372971 0.86 NPY5R (0.41) NPY5RCYP2A6CYP2E1CYP3A4CYP2C9
SCHEMBL7375478 0.84 CYP11B1 (0.43) NPY5RCYP2A6CYP2E1CYP3A4CYP2C9
SCHEMBL28763036 0.75 NPY5R (0.74) NPY5RCYP3A4CYP2C19KDM4ENPC1
Fr-79620 SCHEMBL7370865 0.74 NPY5R (1.00) NPY5RCYP2A6KDM4ENPC1MAPT
SCHEMBL7371445 0.73 NPY5R (0.67) NPY5RMAPTNPSR1L3MBTL1SMPD3
SCHEMBL9634600 0.73 PDE5A (0.40) KDM4ENPC1RAB9AKIT
SCHEMBL27674585 0.73 NPY5R (0.67) NPY5RCYP3A4CYP2C9CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL9838295 0.72 PDE5A (0.41) KDM4ENPC1RAB9AKIT
SCHEMBL7371145 0.72 NPY5R (0.65) NPY5RKDM4ELMNAMAPTNPSR1
SCHEMBL7367119 0.72 MAPK14 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4822805-A ANTIINFLAMMATORY AGENTS, CARDIOTONIC AGENTS, ANTIPLATELET AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-04-18 US disclosed
EP-0257897-A1 Imidazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-03-02 EP disclosed