SCHEMBL7378472

SCHEMBL7378472

CCC(CC)(c1ccccc1)c1cc(O)c(C(c2cccc(NS(=O)(=O)c3ccccc3)c2)C2CC2)c(=O)o1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.36
HTR6 P50406 3/20 0.35
PTGES O14684 1/20 0.35
FABP4 P15090 1/20 0.34
GAA P10253 2/20 0.34
GFER P55789 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
UQCRB P14927 1/20 0.34
HSD17B2 P37059 4/20 0.34
HSD17B1 P14061 3/20 0.34
ALOX12 P18054 1/20 0.34
MAP1LC3B Q9GZQ8 1/20 0.34
MAP1LC3A Q9H492 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
HPGD P15428 1/20 0.33
PDE4B Q07343 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534712 0.92 TGFBR1 (0.35) TGFBR1FABP4GAAGFERAPOBEC3G
SCHEMBL7371141 0.89 TGFBR1 (0.38) TGFBR1HTR6PTGESFABP4GAA
SCHEMBL7368440 0.87 PTGES (0.37) TGFBR1HTR6PTGESFABP4HSD17B2
SCHEMBL7407674 0.86 HTR6 (0.37) TGFBR1HTR6PTGESFABP4GAA
SCHEMBL7367288 0.85 PTGES (0.38) TGFBR1HTR6PTGESFABP4GAA
SCHEMBL7377773 0.85 CYP2C9 (0.36) ALDH1A1
SCHEMBL7367450 0.84 HTR6 (0.38) TGFBR1HTR6PTGESFABP4GAA
SCHEMBL7441063 0.82 KCNK3 (0.36) TGFBR1HTR6PTGESGAAGFER
SCHEMBL7443310 0.82 POLB (0.36) TGFBR1HTR6PTGESGAAGFER
Ethane SCHEMBL7480930 0.81 POLB (0.39) TGFBR1HTR6PTGESGAAGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729465-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP claimed
WO-1995014013-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO claimed
US-6005103-A TREATMENT OF BACTERIAL AND VIRAL INFECTIONS AND DISEASES, INCLUDING AIDS WARNER-LAMBERT COMPANY (US) 1999-12-21 US disclosed
EP-0729465-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014013-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed