SCHEMBL7378592

SCHEMBL7378592

Cn1c(COc2ccc(C#N)cc2)nc2cc(Nc3ccccc3N)ccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.51
RAB9A P51151 6/20 0.46
NPC1 O15118 5/20 0.46
HDAC6 Q9UBN7 1/20 0.46
ALDH1A1 P00352 4/20 0.42
USP2 O75604 1/20 0.42
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 2/20 0.40
GAA P10253 2/20 0.40
F2 P00734 1/20 0.40
ACP1 P24666 1/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.38
RECQL P46063 2/20 0.38
MEN1 O00255 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7379857 0.84 HDAC6 (0.44) PPARGRAB9ANPC1HDAC6ALDH1A1
SCHEMBL6634815 0.74 NPC1 (0.52) RAB9ANPC1HDAC6ALDH1A1LMNA
SCHEMBL7383468 0.73 RAB9A (0.58) PPARGRAB9ANPC1HDAC6ALDH1A1
SCHEMBL7377767 0.72 ALDH1A1 (0.53) PPARGRAB9ANPC1ALDH1A1LMNA
SCHEMBL6635646 0.71 PPARG (0.43) PPARGNPC1HDAC6ALDH1A1USP2
SCHEMBL6636883 0.70 SMN1; SMN2 (0.56) PPARGRAB9ANPC1HDAC6ALDH1A1
SCHEMBL6638614 0.70 F2 (0.43) PPARGRAB9ANPC1HDAC6ALDH1A1
SCHEMBL6781977 0.70 BRPF1 (0.48) PPARGRAB9ANPC1HDAC6ALDH1A1
SCHEMBL14451616 0.70 RAB9A (0.72) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL5901016 0.69 GAA (0.65) RAB9AALDH1A1LMNATP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000050419-A1 SUBSTITUTED BICYCLIC HETEROCYCLES AND THE USE THEREOF AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-08-31 WO disclosed