SCHEMBL7380241

SCHEMBL7380241

Cc1nc(-c2ccc(N3CC(CN4CCN(S(=O)(=O)c5ccc(C(C)(C)C)cc5)CC4)OC3=O)cc2)no1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.46
HSD11B1 P28845 6/20 0.43
POLB P06746 2/20 0.43
ALDH1A1 P00352 2/20 0.41
GBA1 P04062 1/20 0.40
MAPT P10636 2/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39
GRM2 Q14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381271 0.92 SIGMAR1 (0.46) THRBPOLBMAPTLMNATSHR
SCHEMBL7388548 0.90 MAPT (0.45) THRBPOLBALDH1A1GBA1MAPT
SCHEMBL7389136 0.90 SIGMAR1 (0.46) THRBPOLBMAPTLMNATSHR
SCHEMBL7388713 0.89 THRB (0.46) THRBPOLBMAPTLMNATSHR
SCHEMBL7386639 0.89 POLB (0.53) POLBMAPT
SCHEMBL7384895 0.89 THRB (0.44) THRBPOLBALDH1A1MAPTLMNA
SCHEMBL7393478 0.88 TNF (0.44) THRBHSD11B1POLBGBA1MAPT
SCHEMBL7388681 0.88 THRB (0.43) THRBPOLBMAPTLMNATSHR
SCHEMBL7389040 0.86 THRB (0.42) THRBPOLBMAPTLMNATSHR
SCHEMBL7592402 0.86 MAPT (0.46) THRBPOLBMAPTMAOALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056743-A1 BENZAMINE DERIVATIVES MERCK PATENT GmbH (DE) 2000-12-06 EP disclosed
WO-1999031092-A1 BENZAMINE DERIVATIVES MERCK PATENT GMBH (DE) 1999-06-24 WO disclosed